SCHEMBL14239346

SCHEMBL14239346

O=c1c2ccc(-c3ccccn3)cc2nc2n1CC1(CCC2)CC1(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
RAB9A P51151 6/20 0.42
TDP1 Q9NUW8 2/20 0.42
NSD2 O96028 1/20 0.41
ALDH1A1 P00352 4/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
KDM4E B2RXH2 2/20 0.39
USP2 O75604 1/20 0.39
CYP1A2 P05177 1/20 0.39
BCHE P06276 1/20 0.39
CFTR P13569 1/20 0.39
ALOX15 P16050 1/20 0.39
ACHE P22303 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GOPC Q9HD26 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
TGFBR1 P36897 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239321 0.94 NPC1 (0.39) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL14239372 0.88 NPC1 (0.37) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL6923262 0.87 RAB9A (0.46) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL6922046 0.86 NPC1 (0.42) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL14238863 0.83 NPC1 (0.40) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL6922413 0.83 NPC1 (0.43) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL14238900 0.83 NPC1 (0.42) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL14240301 0.82 NPC1 (0.42) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL15834962 0.81 NPC1 (0.40) NPC1RAB9ATDP1NSD2ALDH1A1
SCHEMBL6922198 0.81 ALDH1A1 (0.60) NPC1RAB9ATDP1NSD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed