SCHEMBL14246763

SCHEMBL14246763

CCCc1c(Cc2ccc(Cl)c(Cl)c2)c(=O)[nH]c2cc(OC)cc(OC)c12

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 11/20 0.43
ABCG2 Q9UNQ0 1/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
APLNR P35414 1/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
ALOX5 P09917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15931675 0.92 PDE10A (0.42) PDE10AABCG2PDE3BPDE3AGRIN1
SCHEMBL14317883 0.87 GRIN1 (0.43) PDE10AABCG2PDE3BPDE3AAPLNR
SCHEMBL14317180 0.86 ABCG2 (0.41) PDE10AABCG2PDE3BPDE3A
SCHEMBL15931628 0.83 PDE10A (0.43) PDE10AABCG2PDE3BPDE3A
SCHEMBL15931676 0.79 ABCG2 (0.40) PDE10AABCG2PDE3BPDE3A
SCHEMBL14317220 0.77 GRIN1 (0.46) PDE10APDE3BPDE3AGRIN1GRIN2A
SCHEMBL14317881 0.75 MAPT (0.47) PDE10AABCG2PDE3BPDE3A
SCHEMBL14246722 0.72 PDE10A (0.43) PDE10AABCG2PDE3BPDE3A
SCHEMBL15931626 0.72 ABCG2 (0.44) PDE10AABCG2PDE3BPDE3A
SCHEMBL14246819 0.70 ABCG2 (0.43) PDE10AABCG2PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9334256-B2 Agents and methods for treating ischemic and other diseases NONO INC. (CA) 2016-05-10 US disclosed
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases NONO INC. (CA) 2014-08-07 US disclosed
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases NONO INC. (CA) 2014-08-07 US disclosed
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases NONO INC. (CA) 2014-08-07 US disclosed
EP-2720695-A2 AGENTS AND METHODS FOR TREATING ISCHEMIC AND OTHER DISEASES NoNO Inc. (CA) 2014-04-23 EP disclosed
WO-2012174488-A2 AGENTS AND METHODS FOR TREATING ISCHEMIC AND OTHER DISEASES NONO, INC. (CA) 2012-12-20 WO disclosed
WO-2012174488-A2 AGENTS AND METHODS FOR TREATING ISCHEMIC AND OTHER DISEASES NONO, INC. (CA) 2012-12-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases TRPM7, TRPM8, TRPM5 PDE10A 479/4885ABCG2 2808/4885PDE3B 342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.