SCHEMBL14247238

SCHEMBL14247238

Nc1cc(Br)ccc1NCCC1CCOCC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 6/20 0.44
KDM1A O60341 2/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
CHRM2 P08172 3/20 0.37
CHRM1 P11229 3/20 0.37
CHRM3 P20309 3/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
PRKCQ Q04759 1/20 0.35
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
PRSS1 P07477 2/20 0.34
SCN5A Q14524 1/20 0.34
OPRL1 P41146 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3997126 0.86 AAK1 (0.46) AAK1HDAC1HDAC2
SCHEMBL14247658 0.79 PKM (0.46) PRSS1
SCHEMBL20641725 0.78 NCF1 (0.39) KDM1AMAOAMAOBHDAC1HDAC2
SCHEMBL30437635 0.78 NCF1 (0.39) KDM1AMAOAMAOBHDAC1HDAC2
SCHEMBL14905734 0.76 PRKCQ (0.38) KDM1AMAOAMAOBCHRM2CHRM1
SCHEMBL18172298 0.76 JAK3 (0.38) KDM1AMAOAMAOBCHRM2CHRM1
SCHEMBL2942637 0.75 AAK1 (0.48) AAK1
SCHEMBL2687892 0.75 AAK1 (0.44) AAK1KDM1AMAOAMAOB
SCHEMBL29791971 0.75 AAK1 (0.44) AAK1KDM1AMAOAMAOB
SCHEMBL16035266 0.74 PTGER4 (0.41) AAK1HDAC1HDAC2PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed