SCHEMBL14249396

SCHEMBL14249396

C#Cc1cccc(CF)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
FFAR1 O14842 1/20 0.39
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.35
HDAC8 Q9BY41 1/20 0.32
KDR P35968 1/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3838668 0.82 CA12 (0.44) PTPN1CA12CA1CA2CA9
SCHEMBL30045190 0.78 PNMT (0.48) PTPN1CA12CA1CA2CA9
SCHEMBL29976533 0.78 TRPA1 (0.42) PTPN1CA12CA1CA2CA9
SCHEMBL510419 0.78 FFAR1 (0.46) PTPN1CA12CA1CA2CA9
SCHEMBL4338450 0.78 PNMT (0.48) PTPN1CA12CA1CA2CA9
SCHEMBL30426333 0.78 GLA (0.50) FFAR1GLA
SCHEMBL2795596 0.78 TP53 (0.42) PTPN1CA12CA1CA2CA9
SCHEMBL19806071 0.78 TRPA1 (0.42) PTPN1CA12CA1CA2CA9
SCHEMBL20838047 0.78 CA12 (0.41) PTPN1CA12CA1CA2CA9
SCHEMBL10490628 0.78 GLA (0.35) FFAR1GLAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012172093-A1 DIHYDROINDOLIZINE DERIVATE AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-12-20 WO disclosed