SCHEMBL14251024

SCHEMBL14251024

Fc1cc(Br)cc2ncn(C3CCCOC3)c12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRPS1 P60891 1/20 0.39
JAK1 P23458 4/20 0.34
JAK2 O60674 3/20 0.34
ABL1 P00519 3/20 0.32
OPRM1 P35372 2/20 0.32
OPRK1 P41145 2/20 0.32
JAK3 P52333 2/20 0.30
AURKA O14965 1/20 0.30
PRKCA P17252 1/20 0.30
KDR P35968 1/20 0.30
TYK2 P29597 1/20 0.30
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCND3 P30281 1/20 0.30
CDK6 Q00534 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25924927 0.85 PRPS1 (0.44) PRPS1JAK1JAK2ABL1JAK3
SCHEMBL17042252 0.78 GAA (0.44) JAK1JAK2
SCHEMBL14723562 0.76 CYP2C19 (0.43) PRPS1
SCHEMBL25150851 0.76 BRAF (0.42) ABL1
SCHEMBL14251472 0.75 PRPS1 (0.39) PRPS1JAK1
SCHEMBL14251470 0.75 PRPS1 (0.39) PRPS1JAK1
SCHEMBL14251474 0.75 PRPS1 (0.39) PRPS1JAK1
SCHEMBL31698347 0.74 JAK1 (0.51) PRPS1JAK1JAK2CDK4CCND1
SCHEMBL14325259 0.72 JAK1 (0.38) JAK1JAK2JAK3TYK2CCNC
SCHEMBL21539154 0.72 CDK4 (0.41) PRPS1ABL1OPRM1OPRK1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012172043-A1 PURINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS FOR PREVENTION OR TREATMENT OF BACTERIAL INFECTIONS LABORATOIRE BIODIM (FR) 2012-12-20 WO disclosed
WO-2012172043-A1 PURINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS FOR PREVENTION OR TREATMENT OF BACTERIAL INFECTIONS LABORATOIRE BIODIM (FR) 2012-12-20 WO disclosed