SCHEMBL14257536

SCHEMBL14257536

CNC(=O)/C=C(/C)Nc1ccc(I)cc1F

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 14/20 0.43
MAP2K2 P36507 8/20 0.43
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP2C19 P33261 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HTT P42858 1/20 0.38
PIM1 P11309 1/20 0.37
CAMK2B Q13554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625996 0.80 SMN1; SMN2 (0.48) MAP2K1MAP2K2ALDH1A1HTT
SCHEMBL2650449 0.79 HDAC1 (0.58) MAP2K1MAP2K2HDAC1HDAC6ALDH1A1
SCHEMBL7469020 0.75 ALDH1A1 (0.46) MAP2K1MAP2K2ALDH1A1CYP2C19
SCHEMBL14257414 0.74 NPC1 (0.41) MAP2K1MAP2K2ALDH1A1
SCHEMBL12810857 0.74 NPC1 (0.41) MAP2K1MAP2K2ALDH1A1CYP2C19
SCHEMBL31485290 0.74 MAP2K1 (0.53) MAP2K1MAP2K2ALDH1A1CYP2C19HTT
SCHEMBL12556990 0.74 MAP2K1 (0.46) MAP2K1MAP2K2HDAC1HDAC6ALDH1A1
SCHEMBL22312378 0.73 MAP2K1 (0.42) MAP2K1MAP2K2HDAC1HDAC6HTT
SCHEMBL15058173 0.73 HPGD (0.51) MAP2K1MAP2K2CYP2C19HTTPIM1
SCHEMBL1419646 0.73 KIF11 (0.57) MAP2K1MAP2K2CA1CA2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1894932-A1 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2H-pyrido[2,3-d]pyrimidine derivatives and related compounds for the treatment of cancer Japan Tobacco, Inc. (JP) 2008-03-05 EP disclosed