SCHEMBL1425968

SCHEMBL1425968

C=C(C=CC(N)=O)C(=O)NOS(=O)(=O)CC(C)C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6569861 0.87
SCHEMBL9637961 0.78 TGFBR1 (0.37)
SCHEMBL8592441 0.77
SCHEMBL2153960 0.76
SCHEMBL28379750 0.76 TGFBR1 (0.36)
SCHEMBL10789803 0.74
SCHEMBL1698197 0.71 TSHR (0.39)
SCHEMBL4908429 0.71
SCHEMBL2906578 0.71 CYP2D6 (0.41)
SCHEMBL4913106 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3893833-A1 PERFUME GEL L'OREAL (FR) 2021-10-20 EP claimed
WO-2020120704-A1 PERFUME GEL L'OREAL (FR) 2020-06-18 WO claimed
EP-1570836-A1 Transparent self-tanning gel comprising a hydrosoluble or hydrodispersible polymer of acrylamido 2-methyl propane sulfonic acid L'OREAL (FR) 2005-09-07 EP claimed
EP-0557512-A1 UTILIZATION IN COSMETIC OR TOPICAL APPLICATIONS OF AN AQUEOUS DISPERSION BASED ON ORGANOPOLYSILOXANES AND A CROSSLINKED COPOLYMER OF ACRYLAMIDE/NEUTRALIZED 2-ACRYLAMIDO 2-METHYLPROPANE SULFONIC ACID. OREAL (FR) 1993-09-01 EP claimed
WO-1993005762-A1 UTILIZATION IN COSMETIC OR TOPICAL APPLICATIONS OF AN AQUEOUS DISPERSION BASED ON ORGANOPOLYSILOXANES AND A CROSSLINKED COPOLYMER OF ACRYLAMIDE/NEUTRALIZED 2-ACRYLAMIDO 2-METHYLPROPANE SULFONIC ACID L'OREAL (FR) 1993-04-01 WO claimed
WO-2022129403-A1 COMPOSITION COMPRISING AQUEOUS GELLING AGENTS, SURFACTANTS AND ASCORBIC ACID L'OREAL (FR) 2022-06-23 WO disclosed
EP-3893833-A1 PERFUME GEL L'OREAL (FR) 2021-10-20 EP disclosed
EP-3185843-B1 GEL COMPOSITION AND GEL COMPRISING A UV FILTER OREAL (FR) 2021-08-11 EP disclosed
WO-2020120704-A1 PERFUME GEL L'OREAL (FR) 2020-06-18 WO disclosed
EP-3223778-A1 COSMETIC COMPOSITION COMPRISING A SYNTHETIC PHYLLOSILICATE AND AN ELECTROLYTE AND/OR A POLYELECTROLYTE L'Oréal (FR) 2017-10-04 EP disclosed
EP-3185843-A1 GEL COMPOSITION AND GEL COMPRISING A UV FILTER L'Oréal (FR) 2017-07-05 EP disclosed
EP-2515838-B1 COSMETIC COMPOSITION COMPRISING A JASMONIC ACID DERIVATIVE ORÉAL L (FR) 2016-10-19 EP disclosed
EP-1396256-A2 Cosmetic composition for make-up of keratin fibres L'OREAL (FR) 2004-03-10 EP disclosed
EP-1345919-A2 NOVEL C-GLYCOSIDE DERIVATIVES AND USE THEREOF L'OREAL (FR) 2003-09-24 EP disclosed
EP-1325729-A2 Composition containing a silicone copolymer and an AMPS polymer, and uses thereof, especially in cosmetics L'OREAL (FR) 2003-07-09 EP disclosed
WO-2002051828-A2 NOVEL C-GLYCOSIDE DERIVATIVES AND USE THEREOF L'OREAL (FR) 2002-07-04 WO disclosed
EP-1090629-A1 Aescin and dextran sulfate association L'OREAL (FR) 2001-04-11 EP disclosed
EP-0557512-B1 UTILIZATION IN COSMETIC OR TOPICAL APPLICATIONS OF AN AQUEOUS DISPERSION BASED ON ORGANOPOLYSILOXANES AND A CROSSLINKED COPOLYMER OF ACRYLAMIDE/NEUTRALIZED 2-ACRYLAMIDO 2-METHYLPROPANE SULFONIC ACID OREAL (FR) 1995-12-06 EP disclosed
EP-0557512-A1 UTILIZATION IN COSMETIC OR TOPICAL APPLICATIONS OF AN AQUEOUS DISPERSION BASED ON ORGANOPOLYSILOXANES AND A CROSSLINKED COPOLYMER OF ACRYLAMIDE/NEUTRALIZED 2-ACRYLAMIDO 2-METHYLPROPANE SULFONIC ACID. OREAL (FR) 1993-09-01 EP disclosed
WO-1993005762-A1 UTILIZATION IN COSMETIC OR TOPICAL APPLICATIONS OF AN AQUEOUS DISPERSION BASED ON ORGANOPOLYSILOXANES AND A CROSSLINKED COPOLYMER OF ACRYLAMIDE/NEUTRALIZED 2-ACRYLAMIDO 2-METHYLPROPANE SULFONIC ACID L'OREAL (FR) 1993-04-01 WO disclosed