SCHEMBL14260413

SCHEMBL14260413

COc1ccc(C2(c3ccc(Cl)cc3)CCCCC2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
MAOA P21397 1/20 0.46
CASP1 P29466 2/20 0.46
GAA P10253 1/20 0.46
HSD11B1 P28845 2/20 0.46
KDM4E B2RXH2 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPK1 P28482 1/20 0.44
TSHR P16473 1/20 0.44
SLC6A4 P31645 3/20 0.43
SLC6A3 Q01959 3/20 0.43
SLC6A2 P23975 2/20 0.43
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HDAC1 Q13547 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12893198 0.86 LMNA (0.54) LMNAMAOACASP1GAAL3MBTL1
SCHEMBL12893200 0.86 LMNA (0.54) LMNAMAOACASP1GAAL3MBTL1
SCHEMBL28232465 0.85 LMNA (0.54) LMNAMAOACASP1GAAL3MBTL1
SCHEMBL12893214 0.80 SLC6A4 (0.50) LMNAL3MBTL1MEN1KMT2ATSHR
SCHEMBL17523062 0.77 ESR1 (0.59) LMNACASP1GAAL3MBTL1MEN1
SCHEMBL19268516 0.77 ESR1 (0.59) LMNACASP1GAAL3MBTL1MEN1
SCHEMBL25620272 0.77 ESR1 (0.59) LMNACASP1GAAL3MBTL1MEN1
SCHEMBL29813419 0.76 LMNA (0.49) LMNAMAOACASP1GAAL3MBTL1
SCHEMBL8065672 0.76 LMNA (0.49) LMNAMAOACASP1GAAL3MBTL1
SCHEMBL19863729 0.75 ESR1 (0.58) LMNACASP1GAAL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033894-A2 COMPOUNDS WITH ACTIVITY AT ESTROGEN RECEPTORS ACADIA PHARMACEUTICALS INC. (US) 2008-03-20 WO disclosed
WO-2007056500-A2 COMPOUNDS WITH ACTIVITY AT ESTROGEN RECEPTORS ACADIA PHARMACEUTICALS INC. (US) 2007-05-18 WO disclosed