SCHEMBL14282973

SCHEMBL14282973

BC(=O)N1C[C@H](Oc2cc(-c3ccccc3)nc3cc(OC)ccc23)C[C@H]1C(=O)N[C@]1(C(=O)OCC)CC1CC

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADAM17 P78536 2/20 0.39
TACR3 P29371 8/20 0.38
CTSB P07858 1/20 0.38
CALCRL Q16602 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
ABCC1 P33527 1/20 0.35
ABCC2 Q92887 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14282971 0.90 CTSB (0.40) KDM4EALDH1A1SMN1; SMN2ADAM17TACR3
SCHEMBL14282972 0.90 CTSB (0.40) KDM4EALDH1A1SMN1; SMN2ADAM17TACR3
SCHEMBL12325204 0.87 ADAM17 (0.37) KDM4EALDH1A1SMN1; SMN2ADAM17TACR3
SCHEMBL7945558 0.86 MCL1 (0.40) KDM4EALDH1A1SMN1; SMN2TACR3CTSB
SCHEMBL5692638 0.86 MCL1 (0.40) KDM4EALDH1A1SMN1; SMN2TACR3CTSB
SCHEMBL5692554 0.86 KDM4E (0.39) KDM4EALDH1A1SMN1; SMN2TACR3CTSB
SCHEMBL4979076 0.85 CTSB (0.41) KDM4EALDH1A1SMN1; SMN2ADAM17TACR3
SCHEMBL5692743 0.84 MCL1 (0.40) KDM4EALDH1A1SMN1; SMN2TACR3CTSB
SCHEMBL14307115 0.84 MCL1 (0.40) KDM4EALDH1A1SMN1; SMN2TACR3CTSB
SCHEMBL12325022 0.84 MCL1 (0.39) KDM4EALDH1A1SMN1; SMN2ADAM17TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323447-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-01-29 US disclosed