SCHEMBL14286122

SCHEMBL14286122

CN(C)C(=O)c1cc(-c2cnoc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.48
MAPK1 P28482 3/20 0.46
BCAT1 P54687 1/20 0.42
KMT2A Q03164 3/20 0.38
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 2/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ATM Q13315 1/20 0.34
KDR P35968 1/20 0.34
WNT1 P04628 2/20 0.33
DYRK1A Q13627 2/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
PIM1 P11309 1/20 0.32
PIM2 Q9P1W9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5042374 0.86 BCAT1 (0.45) MAPK1BCAT1NPC1RAB9AKDR
SCHEMBL5047846 0.80 MAPK1 (0.47) POLBMAPK1BCAT1KMT2AGRIN2B
SCHEMBL14286124 0.80 MAPK1 (0.45) POLBMAPK1BCAT1KMT2AGRIN2B
SCHEMBL14600755 0.80 BCAT1 (0.41) POLBMAPK1BCAT1GRIN1GRIN2B
SCHEMBL14600775 0.76 BCAT1 (0.39) POLBBCAT1GRIN1GRIN2BSMN1; SMN2
SCHEMBL14286127 0.74 GSK3B (0.56) MAPK1KMT2ASMN1; SMN2L3MBTL1NPC1
SCHEMBL14286125 0.71 ADORA2A (0.53) POLBKMT2ASMN1; SMN2L3MBTL1NPC1
SCHEMBL4827456 0.70 MAP4K1 (0.45) DYRK1A
SCHEMBL14278769 0.67 GSK3B (0.55) MAPK1KMT2ASMN1; SMN2L3MBTL1NPC1
SCHEMBL14286128 0.67 CCNC (0.41) POLBNPC1RAB9ACCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed