SCHEMBL14286128

SCHEMBL14286128

NC(=O)c1cc(-c2conc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 6/20 0.41
CDK8 P49336 6/20 0.41
PIM1 P11309 2/20 0.39
PIM2 Q9P1W9 2/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
POLB P06746 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PIM3 Q86V86 1/20 0.33
SLC9A1 P19634 1/20 0.33
BTK Q06187 1/20 0.33
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
MAOA P21397 1/20 0.32
BLVRB P30043 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PTGS2 P35354 1/20 0.32
JAK2 O60674 1/20 0.32
CDC7 O00311 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14286138 0.79 GSK3B (0.45)
SCHEMBL14600752 0.77 NPC1 (0.36) PIM1PIM2NPC1RAB9APIM3
SCHEMBL5042374 0.68 BCAT1 (0.45) CCNCCDK8PIM1PIM2NPC1
SCHEMBL14286122 0.67 POLB (0.48) CCNCCDK8PIM1PIM2NPC1
SCHEMBL20792832 0.67 CCNC (0.50) CCNCCDK8PIM1PIM2SLC9A1
SCHEMBL30882693 0.66 MCL1 (0.51) CCNCCDK8PIM1PIM2POLB
SCHEMBL30471591 0.65 CCNC (0.55) CCNCCDK8CDC7
SCHEMBL13175847 0.63 ACMSD (0.50) RAB9AMAOABLVRBHDAC6
SCHEMBL20742135 0.63 CCNC (0.65) CCNCCDK8POLBCDC7
SCHEMBL5047846 0.62 MAPK1 (0.47) NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed