SCHEMBL14288686

SCHEMBL14288686

Cc1cc(C)c(NS(=O)(=O)c2cc(Cl)cc(Cl)c2O)c(C)c1Nc1ccccn1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACLY P53396 16/20 0.51
ALPL P05186 1/20 0.47
BRD4 O60885 1/20 0.47
KDM4E B2RXH2 1/20 0.46
GLA P06280 1/20 0.46
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532884 0.80 ACLY (0.52) ACLYALPLALDH1A1
SCHEMBL8313600 0.78 BRD4 (0.43) BRD4KDM4EGLAMEN1ALDH1A1
SCHEMBL534027 0.77 ACLY (0.55) ACLY
SCHEMBL533156 0.75 ACLY (0.56) ACLY
SCHEMBL532952 0.74 ACLY (0.51) ACLYALPL
SCHEMBL533141 0.73 ACLY (0.63) ACLY
SCHEMBL14288684 0.71 ACLY (0.53) ACLY
SCHEMBL3981809 0.71 ACLY (0.46) ACLYALPL
SCHEMBL532942 0.71 ACLY (0.51) ACLY
SCHEMBL532815 0.70 ACLY (0.53) ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed