SCHEMBL14294451

SCHEMBL14294451

O=c1[nH]ccc2c(Br)c3cccnc3n12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.37
LDHA P00338 1/20 0.36
DAO P14920 1/20 0.36
MAPK8 P45983 1/20 0.35
DYRK1A Q13627 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
AXL P30530 1/20 0.35
HPGD P15428 4/20 0.34
FEN1 P39748 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
MAPT P10636 2/20 0.34
CYP2C9 P11712 1/20 0.34
KDM4E B2RXH2 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
DDB1 Q16531 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13812011 0.82 ACHE (0.37) ACHELDHADAOMAPK8DYRK1A
SCHEMBL14269088 0.73 CDK9 (0.48) ACHELDHAMAPK8DYRK1ACLK4
SCHEMBL4032497 0.71 CDK9 (0.46) ACHEDYRK1AHPGDKDM4ECCNT1
SCHEMBL4034265 0.70 FEN1 (0.35) ACHEFEN1CYP1A2CYP2C19MAPT
SCHEMBL4027865 0.67 MAPK8 (0.43) LDHADAOMAPK8DYRK1ACLK4
SCHEMBL14269066 0.62 MAPK8 (0.41) MAPK8DYRK1ACLK4DYRK1B
SCHEMBL8801077 0.62 AHR (0.48) DAOAXLPIM1
SCHEMBL12165666 0.59 ACHE (0.47) ACHELDHAHPGDFEN1CYP2C19
SCHEMBL25940658 0.59 FEN1 (0.46) DYRK1AHPGDFEN1CYP1A2CYP2C19
SCHEMBL30421286 0.58 AXL (0.53) MAPK8DYRK1ACLK4DYRK1BAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7329666-B2 Derivatives of variolin B PHARMA MAR, S.A. (ES) 2008-02-12 US disclosed