SCHEMBL14304166

SCHEMBL14304166

CCCOc1cc(N)ccc1C(=O)OCCN(C)C

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.80
CYP2D6 P10635 4/20 0.80
SCN1A P35498 4/20 0.80
SCN2A Q99250 4/20 0.80
SCN3A Q9NY46 4/20 0.80
PHLPP2 Q6ZVD8 1/20 0.55
HRH3 Q9Y5N1 5/20 0.52
KCNH2 Q12809 4/20 0.52
MAOA P21397 4/20 0.52
HTR3A P46098 2/20 0.52
HTR2C P28335 2/20 0.52
CHRM2 P08172 1/20 0.52
CHRM3 P20309 1/20 0.52
CHRNA4 P43681 1/20 0.52
CYP3A4 P08684 2/20 0.49
CYP2C19 P33261 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
ALDH1A1 P00352 6/20 0.47
MAPT P10636 2/20 0.47
TSHR P16473 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14304169 0.95 CYP1A2 (0.72) CYP1A2CYP2D6SCN1ASCN2ASCN3A
SCHEMBL22987103 0.89 CYP1A2 (0.78) CYP1A2CYP2D6SCN1ASCN2ASCN3A
Propoxycaine SCHEMBL29353209 0.89 SCN1A (1.00) CYP1A2CYP2D6SCN1ASCN2ASCN3A
Propoxycaine SCHEMBL83073 0.89 SCN1A (1.00) CYP1A2CYP2D6SCN1ASCN2ASCN3A
Propoxycaine SCHEMBL24720 0.88 SCN1A (0.98) CYP1A2CYP2D6SCN1ASCN2ASCN3A
Propoxycaine SCHEMBL1651061 0.86 SCN1A (0.95) CYP1A2CYP2D6SCN1ASCN2ASCN3A
SCHEMBL5925544 0.85 CYP1A2 (0.72) CYP1A2CYP2D6SCN1ASCN2ASCN3A
SCHEMBL10246464 0.84 CYP1A2 (0.70) CYP1A2CYP2D6SCN1ASCN2ASCN3A
Ambucaine SCHEMBL82280 0.84 SCN1A (0.91) CYP1A2CYP2D6SCN1ASCN2ASCN3A
Ambucaine SCHEMBL1007224 0.82 CYP2D6 (0.88) CYP1A2CYP2D6SCN1ASCN2ASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008011539-A2 ANESTHETIC COMPOUNDS PHARMACOFORE, INC. (US) 2008-01-24 WO disclosed