SCHEMBL14304169

SCHEMBL14304169

CCCCOc1cc(N)ccc1C(=O)OCCN(C)C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.72
SCN1A P35498 5/20 0.72
SCN2A Q99250 5/20 0.72
SCN3A Q9NY46 5/20 0.72
CYP2D6 P10635 4/20 0.72
PHLPP2 Q6ZVD8 1/20 0.55
KCNH2 Q12809 5/20 0.52
HRH3 Q9Y5N1 4/20 0.52
MAOA P21397 3/20 0.52
HTR2C P28335 2/20 0.52
CHRM2 P08172 2/20 0.52
CHRM3 P20309 1/20 0.52
CHRNA4 P43681 1/20 0.52
HTR3A P46098 1/20 0.52
TSHR P16473 3/20 0.51
SLC6A3 Q01959 3/20 0.51
SLC6A2 P23975 1/20 0.51
HIF1A Q16665 1/20 0.51
RAD52 P43351 1/20 0.50
LMNA P02545 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14304166 0.95 CYP1A2 (0.80) CYP1A2SCN1ASCN2ASCN3ACYP2D6
SCHEMBL10246464 0.89 CYP1A2 (0.70) CYP1A2SCN1ASCN2ASCN3ACYP2D6
Ambucaine SCHEMBL82280 0.89 SCN1A (0.91) CYP1A2SCN1ASCN2ASCN3ACYP2D6
Ambucaine SCHEMBL1007224 0.88 CYP2D6 (0.88) CYP1A2SCN1ASCN2ASCN3ACYP2D6
SCHEMBL22987103 0.84 CYP1A2 (0.78) CYP1A2SCN1ASCN2ASCN3ACYP2D6
Propoxycaine SCHEMBL29353209 0.84 SCN1A (1.00) CYP1A2SCN1ASCN2ASCN3ACYP2D6
Propoxycaine SCHEMBL83073 0.84 SCN1A (1.00) CYP1A2SCN1ASCN2ASCN3ACYP2D6
Propoxycaine SCHEMBL24720 0.82 SCN1A (0.98) CYP1A2SCN1ASCN2ASCN3ACYP2D6
Propoxycaine SCHEMBL1651061 0.81 SCN1A (0.95) CYP1A2SCN1ASCN2ASCN3ACYP2D6
SCHEMBL13440052 0.81 CYP1A2 (0.58) CYP1A2SCN1ASCN2ASCN3ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008011539-A2 ANESTHETIC COMPOUNDS PHARMACOFORE, INC. (US) 2008-01-24 WO disclosed