SCHEMBL1432043

SCHEMBL1432043

NC(=O)c1nc(Cc2cccnc2)no1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.47
CYP3A4 P08684 2/20 0.44
MEN1 O00255 1/20 0.44
TP53 P04637 1/20 0.44
BLM P54132 1/20 0.44
KMT2A Q03164 1/20 0.44
NAPRT Q6XQN6 1/20 0.44
BMP1 P13497 1/20 0.44
TBXAS1 P24557 6/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
F7 P08709 1/20 0.42
F3 P13726 1/20 0.42
SARM1 Q6SZW1 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
SIRT4 Q9Y6E7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13776650 0.79 MMP2 (0.46) RECQLCYP3A4MEN1KMT2ABMP1
SCHEMBL4497731 0.77 TSHR (0.51) CYP3A4MEN1KMT2ACYP1A2CYP2C9
SCHEMBL13684193 0.76 MMP2 (0.46) TBXAS1CYP1A2MMP2HRH4HRH3
SCHEMBL13728559 0.75 RECQL (0.44) RECQLCYP3A4MEN1TP53BLM
SCHEMBL13728047 0.74 GRM2 (0.47) RECQLCYP3A4MEN1TP53BLM
SCHEMBL4418768 0.74 RECQL (0.47) RECQLCYP3A4MEN1TP53BLM
SCHEMBL4514479 0.74 SRD5A2 (0.48)
SCHEMBL3083749 0.73 L3MBTL1 (0.53) MEN1KMT2AKDM4EMAPTLMNA
SCHEMBL553604 0.72 CHUK (0.53) CYP3A4MEN1KMT2ACYP2C9MAPT
SCHEMBL24658822 0.70 CYP2D6 (0.34) CYP3A4BMP1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300470-A2 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS GABA-A RECEPTOR MODULATORS Sepracor Inc. (US) 2011-03-30 EP disclosed
WO-2009143156-A2 IMIDAZO[1,2-a]PYRIDINE COMPOUNDS SEPRACOR INC. (US) 2009-11-26 WO disclosed