SCHEMBL1432099

SCHEMBL1432099

CC1=CC(N=C=O)(N=C=O)C=C(C)C1c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPK1 P28482 1/20 0.33
HTR2B P41595 1/20 0.33
ALDH1A1 P00352 2/20 0.32
GFER P55789 1/20 0.32
KDM1A O60341 4/20 0.32
MAOA P21397 4/20 0.32
MAOB P27338 4/20 0.32
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GAA P10253 3/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
SLC9A1 P19634 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7115170 0.78
SCHEMBL3679608 0.71 MAOA (0.43) MAPTLMNATP53CYP1A2CYP3A4
SCHEMBL9224978 0.70 KDM1A (0.47) MAPTLMNATP53CYP1A2CYP3A4
SCHEMBL3412624 0.68
SCHEMBL8734945 0.67 MAPT (0.34) MAPTLMNATP53CYP1A2CYP3A4
SCHEMBL3223717 0.61 CYP1A2 (0.42) MAPTLMNATP53CYP1A2CYP3A4
SCHEMBL9250732 0.61 CYP1A2 (0.42) MAPTLMNATP53CYP1A2CYP3A4
SCHEMBL9281441 0.59 MAPT (0.46) MAPTLMNATP53CYP1A2CYP3A4
Methylamine SCHEMBL27321608 0.58 CYP3A4 (0.48) MAPTLMNACYP1A2CYP3A4MAPK1
SCHEMBL20955661 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090053490-A1 Highly Filled Composite Materials CLAUSI ROBERT N 2009-02-26 US claimed
EP-1991608-A1 HIGHLY FILLED COMPOSITE MATERIALS Clausi, Robert N. (CA) 2008-11-19 EP claimed
WO-2007095730-A1 HIGHLY FILLED COMPOSITE MATERIALS CLAUSI ROBERT N (CA) 2007-08-30 WO claimed
CN-111479837-B Flexible packaging material for preserving food freshness 陶氏环球技术有限责任公司 2022-08-23 CN disclosed
US-11214648-B2 Spray foam building insulation for exterior applications DILORETO SALVATORE A (CA) 2022-01-04 US disclosed
US-20210115184-A1 SPRAY FOAM BUILDING INSULATION FOR EXTERIOR APPLICATIONS DILORETO SALVATORE A (CA) 2021-04-22 US disclosed
CN-111479837-A Flexible packaging material for preserving food freshness 陶氏环球技术有限责任公司 2020-07-31 CN disclosed
EP-3548560-A1 SPRAY FOAM BUILDING INSULATION FOR EXTERIOR APPLICATIONS Diloreto, Salvatore Anthony (CA) 2019-10-09 EP disclosed
US-10086531-B2 Process for producing resilient wood particleboard, MDF and HDF CLAUSI ROBERT N (CA) 2018-10-02 US disclosed
US-10012343-B2 Pallet stacking board construction RIVER ROCK INDUSTRIES CORP. (CA) 2018-07-03 US disclosed
WO-2018098570-A1 SPRAY FOAM BUILDING INSULATION FOR EXTERIOR APPLICATIONS DILORETO SALVATORE A (CA) 2018-06-07 WO disclosed
US-20090326088-A1 Pre-Reacted Isocyanate Product Elastochem Specialty Chemicals Inc. (CA) 2009-12-31 US disclosed
US-20090324924-A1 Process and System For Insulating A Surface Using A Polyurethane Foam Made From A Pre-Reacted Isocyanate GUARDIAN BUILDING PRODUCTS (US) 2009-12-31 US disclosed
EP-2126234-A1 POLYURETHANE FOAM BATT INSULATION Diloreto, Salvatore Anthony (CA) 2009-12-02 EP disclosed
US-20090053490-A1 Highly Filled Composite Materials CLAUSI ROBERT N 2009-02-26 US disclosed
EP-1991608-A1 HIGHLY FILLED COMPOSITE MATERIALS Clausi, Robert N. (CA) 2008-11-19 EP disclosed
WO-2008106801-A1 POLYURETHANE FOAM BATT INSULATION DILORETO SALVATORE ANTHONY (CA) 2008-09-12 WO disclosed
WO-2007095730-A1 HIGHLY FILLED COMPOSITE MATERIALS CLAUSI ROBERT N (CA) 2007-08-30 WO disclosed
WO-2005034781-A1 DEVICES AND METHODS FOR SPINE REPAIR PROMETHEAN SURGICAL DEVICES LLC (US) 2005-04-21 WO disclosed
US-4367259-A A POLYETHERURETHANE COPOLYMER BINDER CONTAINING SOUND DEADENING PARTICLES W. R. GRACE & CO. (US) 1983-01-04 US disclosed