SCHEMBL14336403

SCHEMBL14336403

COc1cc(N)ccc1S(=O)(=O)/N=C/N(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 3/20 0.39
MAPT P10636 3/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
RAPGEF3 O95398 1/20 0.37
PKM P14618 1/20 0.36
KDM4E B2RXH2 2/20 0.36
TRPV4 Q9HBA0 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
CYP19A1 P11511 3/20 0.35
NQO2 P16083 1/20 0.35
NR4A1 P22736 1/20 0.35
F2 P00734 2/20 0.34
PRSS1 P07477 2/20 0.34
PRSS2 P07478 2/20 0.34
PRSS3 P35030 2/20 0.34
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151649 0.79 HTT (0.48) GAALMNAALDH1A1HTTPKM
SCHEMBL5151645 0.79 HTT (0.48) GAALMNAALDH1A1HTTPKM
SCHEMBL14336285 0.79 HTT (0.48) GAALMNAALDH1A1HTTPKM
SCHEMBL24686355 0.78 GAA (0.49) GAALMNAALDH1A1MAPTTSHR
SCHEMBL27715369 0.77 LMNA (0.42) GAALMNAALDH1A1MAPTTSHR
SCHEMBL19551921 0.77 LMNA (0.44) GAALMNAALDH1A1MAPTKDM4E
SCHEMBL19551919 0.77 LMNA (0.44) GAALMNAALDH1A1MAPTKDM4E
SCHEMBL29718844 0.77 LMNA (0.44) GAALMNAALDH1A1MAPTKDM4E
SCHEMBL10642047 0.75 GAA (0.54) GAALMNATSHRMAPK1HTT
SCHEMBL10642042 0.75 GAA (0.54) GAALMNATSHRMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312225-B2 Macrocyclic pyrimidines, their production and use as pharmaceutical agents BAYER SCHERING PHARMA AG (DE) 2007-12-25 US disclosed