SCHEMBL14345747

SCHEMBL14345747

Cc1c2n(cnc1=O)CCc1c-2[nH]c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 13/20 0.51
CYP1B1 Q16678 13/20 0.51
CYP1A2 P05177 13/20 0.51
KDM4E B2RXH2 4/20 0.51
HSD17B10 Q99714 3/20 0.51
POLB P06746 2/20 0.51
NPC1 O15118 2/20 0.51
ALDH1A1 P00352 2/20 0.51
TSHR P16473 2/20 0.51
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
PDE5A O76074 2/20 0.51
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51
CYP3A4 P08684 1/20 0.51
PKM P14618 1/20 0.51
PTGS1 P23219 1/20 0.51
PTGS2 P35354 1/20 0.51
THPO P40225 1/20 0.51
MTOR P42345 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14345741 0.83 CYP1A2 (0.57) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL14345950 0.83 CYP1A2 (0.49) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL14346052 0.80 CYP1A1 (0.60) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL14345736 0.75 ALDH1A1 (0.47) CYP1A2KDM4EHSD17B10ALDH1A1TSHR
SCHEMBL14345725 0.75 CYP1A1 (0.57) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL14345705 0.74 BCHE (0.50) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL14345951 0.72 CYP1A2 (0.57) CYP1A1CYP1B1CYP1A2KDM4EPOLB
SCHEMBL14345847 0.71 CYP1A1 (0.58) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL1311759 0.68 KDM4E (0.64) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10
SCHEMBL2457583 0.68 KDM4E (0.47) CYP1A1CYP1B1CYP1A2KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007138081-A1 PYRIMIDINO[1',6'-1,2]PYRIDO[3,4-b]INDOLE DERIVATIVES AND THEIR THERAPEUTIC USAGE FOURTILLAN (FR) 2007-12-06 WO disclosed