Rivoglitazone

Rivoglitazone

SCHEMBL143498

COc1ccc2nc(COc3ccc(CC4SC(=O)NC4=O)cc3)n(C)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARG

The experimentally established mechanism targets of Rivoglitazone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPARG known ✓ P37231 12/20 1.00
ESRRA P11474 1/20 0.73
FFAR1 O14842 11/20 0.63
PPARA Q07869 6/20 0.63
MPC2 O95563 1/20 0.54
CYP2C8 P10632 1/20 0.54
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rivoglitazone SCHEMBL5319250 1.00 PPARG (1.00) PPARGESRRAFFAR1PPARAMPC2
Rivoglitazone SCHEMBL2906120 1.00 PPARG (1.00) PPARGESRRAFFAR1PPARAMPC2
Rivoglitazone SCHEMBL1592290 0.99 PPARG (0.98) PPARGESRRAFFAR1PPARAMPC2
Rivoglitazone SCHEMBL6064788 0.99 PPARG (0.98) PPARGESRRAFFAR1PPARAMPC2
Rivoglitazone SCHEMBL4885815 0.96 PPARG (0.91) PPARGESRRAFFAR1PPARAMPC2
SCHEMBL6543624 0.95 PPARG (0.90) PPARGESRRAFFAR1PPARAMPC2
Hydrochloric Acid SCHEMBL6544473 0.94 PPARG (0.88) PPARGESRRAFFAR1PPARAMPC2
SCHEMBL15730390 0.94 PPARG (0.88) PPARGESRRAFFAR1PPARAMPC2
SCHEMBL6896700 0.93 PPARG (0.86) PPARGESRRAFFAR1PPARAMPC2
SCHEMBL14168935 0.92 PPARG (0.84) PPARGESRRAFFAR1PPARAMPC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1900 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360215-A1 PHARMACEUTICAL COMBINATIONS AND METHODS FOR PREVENTING OR TREATING NEURODEGENERATIVE DISEASES YUH CHIOU HWA (US) 2025-11-27 US claimed
US-20250332101-A1 Composition CORDEIRO MARIA FRANCESCA (GB) 2025-10-30 US claimed
EP-4640701-A2 GLUCAGON LIKE PEPTIDE 1 (GLP-1) FUSION PEPTIDE COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE CONJUGATES AND USES THEREOF Janssen Sciences Ireland Unlimited Company (IE) 2025-10-29 EP claimed
US-20250281507-A1 METHODS OF TREATING NEPHROTIC SYNDROME THE RESEARCH INSTITUTE AT NATIONWIDE CHILDREN’S HOSPITAL 2025-09-11 US claimed
US-20250221962-A1 FABP4 AS A THERAPEUTIC TARGET IN SKIN DISEASES TICURE LTD (IL) 2025-07-10 US claimed
WO-2025136060-A1 CULTURE MEDIUM COMPOSITION FOR TRANSDIFFERENTIATION OF MUSCLE STEM CELLS INTO ADIPOCYTES, AND METHOD FOR PRODUCING CULTURED MEAT BY USING SAME 한화솔루션 주식회사 2025-06-26 WO claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250082781-A1 METHODS OF LOWERING BLOOD GLUCOSE AND TREATING TYPE 2 DIABETES BY ACTIVATION OF PDE4D3 SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2025-03-13 US claimed
EP-4520343-A2 GLUCAGON LIKE PEPTIDE 1 (GLP1)-GROWTH DIFFERENTIATION FACTOR 15 (GDF15) FUSION PROTEINS AND USES THEREOF Janssen Sciences Ireland Unlimited Company (IE) 2025-03-12 EP claimed
WO-2025049710-A1 PHARMACEUTICAL COMPOSITION FOR USE IN THE DISEASE TREATMENTS ACLIPSE TWO INC. (US) 2025-03-06 WO claimed
EP-0796618-B1 Treatment and prophylaxis of pancreatitis SANKYO CO (JP) 2002-01-30 EP claimed
EP-0753298-B1 Synergistic combination comprising an insulin sensitizer and a HMG-CoA reductase inhibitor for treating arteriosclerosis SANKYO CO (JP) 2001-11-21 EP claimed
EP-0745600-B1 Benzimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-10-24 EP claimed
US-6159997-A Treatment of arteriosclerosis and xanthoma SANKYO COMPANY, LIMITED (JP) 2000-12-12 US claimed
US-6150371-A WITH THE EXCEPTION OF TYPE I DIABETES; INHIBITS INVASION OF ORGAN TISSUE BY CYTOTOXIC LYMPHOCYTES; ADMINISTERING TO A MAMMAL AN ANTIAUTOIMMUNE DISEASE AGENT BEING AN INSULIN RESISTANCE REDUCING AGENT, ANTIDIABETIC, E.G., TROGLITAZONE SANKYO COMPANY, LIMITED (JP) 2000-11-21 US claimed
WO-2000041690-A1 USE OF THIAZOLIDINEDIONES TO AMELIORATE THE ADVERSE CONSEQUENCES OF MYOCARDIAL ISCHEMIA ON MYOCARDIAL FUNCTION AND METABOLISM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-07-20 WO claimed
EP-0919232-A1 Composition for use in the treatment and prevention of hyperuricemia Sankyo Company Limited (JP) 1999-06-02 EP claimed
EP-0796618-A1 Treatment and prophylaxis of pancreatitis SANKYO COMPANY LIMITED (JP) 1997-09-24 EP claimed
EP-0753298-A1 Synergistic combination comprising an insulin sensitizer and a HMG-CoA reductase inhibitor for treating arteriosclerosis SANKYO COMPANY LIMITED (JP) 1997-01-15 EP claimed
EP-0745600-A1 Benzimidazole derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1996-12-04 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250082781-A1 METHODS OF LOWERING BLOOD GLUCOSE AND TREATING TYPE 2 DIABETES BY ACTIVATION OF PDE4D3 PDE4D, PDE4A, PDE4B PPARG 129/4885ESRRA 1192/4885FFAR1 1346/4885
US-20250281507-A1 METHODS OF TREATING NEPHROTIC SYNDROME PPARA, PPARG, PPARD PPARG 2/4885ESRRA 217/4885FFAR1 131/4885
US-20250221962-A1 FABP4 AS A THERAPEUTIC TARGET IN SKIN DISEASES FABP4, FABP2, FABP1 PPARG 46/4885ESRRA 3040/4885FFAR1 392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.