SCHEMBL14356409

SCHEMBL14356409

O=C(NCc1ccccc1)c1ccccc1-n1cccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.66
ALDH1A1 P00352 1/20 0.64
APEX1 P27695 1/20 0.61
CYP2C19 P33261 2/20 0.59
CYP2C9 P11712 1/20 0.59
HPGD P15428 3/20 0.58
GAA P10253 2/20 0.58
LMNA P02545 2/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
METAP2 P50579 1/20 0.56
CHRNB2 P17787 1/20 0.56
CHRNB4 P30926 1/20 0.56
CHRNA3 P32297 1/20 0.56
CHRNA4 P43681 1/20 0.56
TP53 P04637 1/20 0.54
GLA P06280 1/20 0.54
CYP1A2 P05177 1/20 0.54
NSD2 O96028 2/20 0.52
SGMS2 Q8NHU3 1/20 0.52
USP2 O75604 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11901003 0.81 KMT2A (0.89) KMT2AAPEX1CYP2C19CYP2C9HPGD
SCHEMBL31680569 0.81 KMT2A (0.89) KMT2AAPEX1CYP2C19CYP2C9HPGD
SCHEMBL8635709 0.80 KMT2A (1.00) KMT2AAPEX1CYP2C19CYP2C9HPGD
SCHEMBL1984940 0.80 KMT2A (1.00) KMT2AAPEX1CYP2C19CYP2C9HPGD
SCHEMBL23708473 0.79 KMT2A (0.62) KMT2AALDH1A1APEX1CYP2C19HPGD
SCHEMBL14738627 0.79 KMT2A (0.62) KMT2AALDH1A1APEX1CYP2C19HPGD
SCHEMBL6387047 0.78 ALDH1A1 (0.69) KMT2AALDH1A1CYP2C19CYP2C9GAA
SCHEMBL1520747 0.78 ALDH1A1 (1.00) KMT2AALDH1A1CYP2C19CYP2C9GAA
SCHEMBL17481995 0.77 KMT2A (0.51) KMT2AALDH1A1APEX1CYP2C19CYP2C9
SCHEMBL974278 0.76 ALDH1A1 (0.71) KMT2AALDH1A1CYP2C19CYP2C9GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291621-B2 Substituted biaryl amides C5a receptor modulators NEUROGEN CORPORATION (US) 2007-11-06 US disclosed
US-7291621-B2 Substituted biaryl amides C5a receptor modulators NEUROGEN CORPORATION (US) 2007-11-06 US disclosed