SCHEMBL143620

SCHEMBL143620

COC(=O)c1cccc(C(=O)c2c(C)c(OC)c3ccccn23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.48
ALDH1A1 P00352 8/20 0.47
KMT2A Q03164 6/20 0.43
MEN1 O00255 4/20 0.43
HPGD P15428 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MAPT P10636 6/20 0.43
LMNA P02545 4/20 0.43
GAA P10253 3/20 0.43
NPC1 O15118 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ATM Q13315 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
POLB P06746 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722235 0.89 HTT (0.52) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL3608384 0.89 HTT (0.51) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL4511548 0.86 HTT (0.48) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL321257 0.83 MAPT (0.43) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL145768 0.80 HTT (0.55) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL2519397 0.79 NPC1 (0.46) HTTALDH1A1KMT2AMEN1MAPT
SCHEMBL6218948 0.79 HTT (0.51) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL320712 0.79 HTT (0.51) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL6217961 0.79 NPC1 (0.46) HTTALDH1A1KMT2AMEN1HPGD
Hydrochloric Acid SCHEMBL3611393 0.79 NPC1 (0.46) HTTALDH1A1KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8034828-B2 Use of FGF inhibiting substituted 1,2,3 indolizine derivatives in the preparation of medicaments which can be used to treat diseases linked to pathological choroidal angiogenesis SANOFI-AVENTIS (FR) 2011-10-11 US claimed
EP-1713543-B1 USE OF SUBSTITUTED 1,2,3 INDOLIZINE DERIVATIVES FOR TREATING DISEASES ASSOCIATED WITH A PATHOLOGICAL ANGIOGENESIS SANOFI AVENTIS (FR) 2009-11-11 EP claimed
US-20090030034-A1 USE OF FGF INHIBITING SUBSTITUTED 1,2,3 INDOLIZINE DERIVATIVES IN THE PREPARATION OF MEDICAMENTS WHICH CAN BE USED TO TREAT DISEASES LINKED TO PATHOLOGICAL CHOROIDAL ANGIOGENESIS SANOFI-AVENTIS (FR) 2009-01-29 US claimed
US-20140221455-A1 DIFFERENTIATION MODULATING AGENTS AND USES THEREFOR Verva Pharmaceuticals, Inc. (AU) 2014-08-07 US disclosed
US-20120059047-A1 DIFFERENTIATION MODULATING AGENTS AND USES THEREFOR VERVA PHARMACEUTICALS PTY LTD (AU) 2012-03-08 US disclosed
US-8034828-B2 Use of FGF inhibiting substituted 1,2,3 indolizine derivatives in the preparation of medicaments which can be used to treat diseases linked to pathological choroidal angiogenesis SANOFI-AVENTIS (FR) 2011-10-11 US disclosed
US-20090030034-A1 USE OF FGF INHIBITING SUBSTITUTED 1,2,3 INDOLIZINE DERIVATIVES IN THE PREPARATION OF MEDICAMENTS WHICH CAN BE USED TO TREAT DISEASES LINKED TO PATHOLOGICAL CHOROIDAL ANGIOGENESIS SANOFI-AVENTIS (FR) 2009-01-29 US disclosed
US-20050282733-A1 Differentiation modulating agents and uses therefor VERVA PHARMACEUTICALS PTY LTD (AU) 2005-12-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059047-A1 DIFFERENTIATION MODULATING AGENTS AND USES THEREFOR FGF1, FABP4, FGF2 HTT 3582/4885ALDH1A1 1103/4885KMT2A 3024/4885
US-20090030034-A1 USE OF FGF INHIBITING SUBSTITUTED 1,2,3 INDOLIZINE DERIVATIVES IN THE PREPARATION OF MEDICAMENTS WHICH CAN BE USED TO TREAT DISEASES LINKED TO PATHOLOGICAL CHOROIDAL ANGIOGENESIS FGF1, FGF2, FGFR1 HTT 3824/4885ALDH1A1 594/4885KMT2A 3872/4885
US-20050282733-A1 Differentiation modulating agents and uses therefor FGF1, FABP4, FGF2 HTT 3582/4885ALDH1A1 1103/4885KMT2A 3024/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.