SCHEMBL14368290

SCHEMBL14368290

CCn1c(Cn2ccnc2-c2cc(F)ccc2F)nc2cc(C)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.40
RPS6KA5 O75582 1/20 0.37
MAPT P10636 4/20 0.35
GAA P10253 3/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
GRIN2B Q13224 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
THRB P10828 1/20 0.35
PABPC1 P11940 1/20 0.35
HPGD P15428 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3060330 0.95 RPS6KA5 (0.41) RPS6KA5MAPTGAACYP11B1CYP11B2
SCHEMBL3065544 0.91 TBXA2R (0.39) RPS6KA5MAPTCYP11B1CYP11B2KMT2A
SCHEMBL3060709 0.90 KDM4E (0.45) RPS6KA5MAPTGAACYP11B1CYP11B2
SCHEMBL3062446 0.89 CYP11B1 (0.36) RPS6KA5MAPTGAACYP11B1CYP11B2
SCHEMBL3054829 0.88 CNR2 (0.38) RPS6KA5GRIN2BMEN1KMT2AKDM4E
SCHEMBL3059727 0.88 RPS6KA5 (0.34) RPS6KA5MAPTGAACYP11B1CYP11B2
SCHEMBL3060160 0.88 S1PR1 (0.36) RPS6KA5MAPTGAACYP11B1CYP11B2
SCHEMBL3055159 0.87 THRB (0.52) NLRP3MAPTGAAMEN1KMT2A
SCHEMBL3068783 0.87 MAPT (0.43) NLRP3RPS6KA5MAPTGAAMEN1
SCHEMBL3065422 0.87 ALDH1A1 (0.41) GAAALDH1A1KDM4EHPGDTBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7300945-B2 Benzimidazole and pyridylimidazole derivatives NEUROGEN CORPORATION (US) 2007-11-27 US disclosed