SCHEMBL1438600

SCHEMBL1438600

CCCCc1ccc(COc2ccc(C3CN(CCC(=O)O)CCO3)c(C)c2)cc1.Cc1ccc(COc2ccc(C3CN(CCC(=O)O)CCO3)c(C)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.43
FFAR1 O14842 6/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
KDM2B Q8NHM5 1/20 0.39
FFAR4 Q5NUL3 4/20 0.38
S1PR1 P21453 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
DRD3 P35462 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1438239 0.97 HRH3 (0.45) HRH3FFAR1GRIN1GRIN2BKDM2B
SCHEMBL1438821 0.93 HRH3 (0.42) HRH3FFAR1KDM2BS1PR1
SCHEMBL1438604 0.93 HRH3 (0.41) HRH3FFAR1GRIN1GRIN2BKDM2B
SCHEMBL1438554 0.92 THRB (0.43) HRH3FFAR1GRIN1GRIN2BKDM2B
SCHEMBL15484527 0.88 DRD3 (0.46) HRH3GRIN1GRIN2BKDM2BDRD3
SCHEMBL1439048 0.88 HRH3 (0.41) HRH3GRIN1GRIN2BKDM2BDRD3
SCHEMBL1438100 0.87 EGFR (0.48) FFAR1GRIN1GRIN2BKDM2BFFAR4
SCHEMBL1437924 0.87 FFAR1 (0.44) HRH3FFAR1GRIN1GRIN2BS1PR1
SCHEMBL1438702 0.87 S1PR5 (0.48) FFAR1GRIN1GRIN2BKDM2BS1PR1
SCHEMBL1438072 0.86 GRIN1 (0.45) HRH3FFAR1GRIN1GRIN2BFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473490-A1 (THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS Abbott Healthcare Products B.V. (NL) 2012-07-11 EP claimed
WO-2011023795-A1 (THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS ABBOTT HEALTHCARE PRODUCTS B.V. (NL) 2011-03-03 WO claimed