SCHEMBL1438604

SCHEMBL1438604

CCCCc1ccc(COc2ccc(C3CN(CCC(=O)OC(=O)CCN4CCOC(c5ccc(OCc6ccc(C)cc6)cc5C)C4)CCO3)c(C)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.41
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
DRD3 P35462 4/20 0.37
KDM2B Q8NHM5 1/20 0.37
SMPD1 P17405 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAOB P27338 3/20 0.36
THRB P10828 2/20 0.36
THRA P10827 1/20 0.36
ACHE P22303 1/20 0.36
FFAR1 O14842 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1438600 0.93 HRH3 (0.43) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL1439048 0.90 HRH3 (0.41) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL1438239 0.90 HRH3 (0.45) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL15484527 0.87 DRD3 (0.46) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL1438485 0.86 NPC1 (0.39) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL1438821 0.85 HRH3 (0.42) HRH3KDM2BNPC1GAAHPGD
SCHEMBL1437865 0.85 PSEN1 (0.41) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL1438554 0.84 THRB (0.43) HRH3GRIN1GRIN2BDRD3KDM2B
SCHEMBL1438183 0.80 DRD4 (0.40) HRH3GRIN1GRIN2BSMPD1NPC1
SCHEMBL1438100 0.80 EGFR (0.48) GRIN1GRIN2BKDM2BFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473490-A1 (THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS Abbott Healthcare Products B.V. (NL) 2012-07-11 EP claimed
WO-2011023795-A1 (THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS ABBOTT HEALTHCARE PRODUCTS B.V. (NL) 2011-03-03 WO claimed