SCHEMBL14386355

SCHEMBL14386355

C=NN(/C(=N\N)N1CCN(C(=O)C(=O)c2c[nH]c3c(-c4cc(C(=O)NCCN5CCOCC5)[nH]n4)ncc(F)c23)CC1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 3/20 0.37
BCL3 P20749 4/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
CCNT1 O60563 2/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CDK9 P50750 2/20 0.34
HSD17B10 Q99714 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BACE1 P56817 1/20 0.34
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14386113 0.95 SMYD2 (0.34) KDM4EHSD17B10
SCHEMBL14385555 0.91 CYP2C9 (0.41) KDM5BBCL3HPGDKDM4EALDH1A1
SCHEMBL14386354 0.91 KDM4E (0.34) HPGDKDM4EALDH1A1SMN1; SMN2CYP1A2
SCHEMBL14386112 0.87 ALDH1A1 (0.34) ALDH1A1SMN1; SMN2GAA
SCHEMBL2629097 0.86 CYP2C9 (0.42) KDM5BBCL3HPGDKDM4EALDH1A1
SCHEMBL14385644 0.86 CYP2C9 (0.42) ALDH1A1CYP1A2CYP2C19
SCHEMBL14385558 0.85 CYP2C9 (0.41) HPGDKDM4EALDH1A1HSD17B10CYP1A2
SCHEMBL14385667 0.83 HPGDS (0.36) KMT2ACYP1A2CYP2C19
SCHEMBL14385669 0.83 CYP2C9 (0.33) CYP1A2CYP2C19
SCHEMBL15204074 0.82 KDM5B (0.40) KDM5BBCL3HPGDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007127635-A2 DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-08 WO disclosed