SCHEMBL14396751

SCHEMBL14396751

CCOC(=O)c1ccc(CN(CCCCC(=O)OC)CCc2ccccc2OCc2ccc(-c3ccc(OC)cc3)cc2F)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CETP P11597 5/20 0.39
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ACHE P22303 1/20 0.36
MEP1B Q16820 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
S1PR1 P21453 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6401258 0.94 LPAR1 (0.37) CETPLMNAHDAC1HDAC6ACHE
SCHEMBL5275145 0.85 LPAR1 (0.43) MEP1BS1PR1
SCHEMBL13009752 0.85 MAPT (0.42) LMNAACHEMEN1KMT2ASMN1; SMN2
SCHEMBL13009651 0.82 ABCB1 (0.46) LMNAMEP1BMEN1KMT2AMAPT
SCHEMBL13009864 0.82 BCHE (0.42) LMNAACHEMEN1KMT2ASMN1; SMN2
SCHEMBL13009801 0.81 CETP (0.44) CETPLMNATP53LTB4R2ACHE
SCHEMBL13009787 0.81 LMNA (0.38) CETPLMNATP53ACHEMEN1
SCHEMBL13009903 0.81 MTNR1B (0.42) MEP1BMEN1KMT2ASMN1; SMN2MAPT
SCHEMBL13009871 0.80 MAPT (0.39) CETPLMNATP53ACHEMEN1
SCHEMBL13009844 0.80 MAPT (0.40) CETPLMNAACHEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368301-B1 SIDE-CHAIN HALOGENATED AMINO CARBOXYLIC ACID DERIVATIVES AS MEDICAMENTS FOR TREATING CARDIOVASCULAR DISEASES BAYER HEALTHCARE AG (DE) 2007-10-31 EP disclosed