SCHEMBL14399552

SCHEMBL14399552

CCc1ccc(C(=O)NCCN(C)CC)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
LMNA P02545 2/20 0.54
SLC22A2 O15244 1/20 0.54
SLC22A1 O15245 1/20 0.54
TSHR P16473 1/20 0.54
ACHE P22303 1/20 0.54
MAPK1 P28482 1/20 0.54
CYP2C19 P33261 1/20 0.54
TMEM97 Q5BJF2 5/20 0.53
SIGMAR1 Q99720 5/20 0.53
PLK1 P53350 1/20 0.53
BLM P54132 2/20 0.52
PMP22 Q01453 1/20 0.52
NFKB1 P19838 1/20 0.50
KCNH2 Q12809 1/20 0.50
OPRK1 P41145 3/20 0.49
OPRM1 P35372 1/20 0.49
POLB P06746 2/20 0.49
CYP3A4 P08684 1/20 0.49
THRB P10828 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10076245 0.87 ALDH1A1 (0.66) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL12845484 0.86 LMNA (0.72) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL11966131 0.86 LMNA (0.58) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL17688292 0.85 ALDH1A1 (0.62) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL14370083 0.83 TMEM97 (0.59) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL14947438 0.81 HPGD (0.67) ALDH1A1TMEM97SIGMAR1PLK1POLB
SCHEMBL8128025 0.81 ALDH1A1 (0.50) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL8404684 0.80 ALDH1A1 (0.56) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL6360077 0.80 PLK1 (0.63) ALDH1A1LMNAMAPK1PLK1
SCHEMBL3322603 0.80 KDM4E (0.69) ALDH1A1LMNASLC22A2SLC22A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279469-B2 Diaminotriazoles useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-09 US disclosed