SCHEMBL1439986

SCHEMBL1439986

O=c1[nH]c2cc(F)c(Cl)cc2[nH]1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.63
TDP1 Q9NUW8 1/20 0.63
GRIA1 P42261 8/20 0.50
GRIN2D O15399 4/20 0.50
GRIN3B O60391 4/20 0.50
GRIN1 Q05586 4/20 0.50
GRIN2A Q12879 4/20 0.50
GRIN2B Q13224 4/20 0.50
GRIN2C Q14957 4/20 0.50
GRIN3A Q8TCU5 4/20 0.50
MAPT P10636 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
THPO P40225 1/20 0.50
GRIA2 P42262 1/20 0.50
GRIA3 P42263 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL462766 0.86 GRIN2D (0.70) ALDH1A1TDP1GRIA1GRIN2DGRIN3B
SCHEMBL3786399 0.83 PDE3B (0.50) ALDH1A1TDP1GRIA1GRIN2DGRIN3B
SCHEMBL640124 0.83 GRIA1 (0.70) ALDH1A1GRIA1GRIN2DGRIN3BGRIN1
SCHEMBL8137325 0.82 ALDH1A1 (0.47) ALDH1A1TDP1GRIA1GRIN2DGRIN3B
SCHEMBL29909816 0.82 ALDH1A1 (0.47) ALDH1A1TDP1GRIA1GRIN2DGRIN3B
SCHEMBL17432052 0.77 ALDH1A1 (1.00) ALDH1A1TDP1GRIA1GRIN2DGRIN3B
SCHEMBL1115539 0.73 GRIA1 (0.50) ALDH1A1GRIA1GRIN2DGRIN3BGRIN1
SCHEMBL22725084 0.73 MAPT (0.42) ALDH1A1TDP1GRIN2DGRIN3BGRIN1
SCHEMBL17758383 0.73 PDE3B (0.41) ALDH1A1TDP1GRIA1GRIN2DGRIN3B
SCHEMBL31748445 0.73 MAPT (0.42) ALDH1A1TDP1GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011023812-A1 MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 (MPGES1) INHIBITORS NOVASAID AB (SE) 2011-03-03 WO disclosed
WO-2011023812-A1 MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 (MPGES1) INHIBITORS NOVASAID AB (SE) 2011-03-03 WO disclosed