SCHEMBL22725084

SCHEMBL22725084

O=c1[nH]c2cc(F)c(Br)cc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.42
ALDH1A1 P00352 5/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
PAX8 Q06710 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
ABL1 P00519 1/20 0.38
NTRK1 P04629 1/20 0.38
FYN P06241 1/20 0.38
RET P07949 1/20 0.38
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31748445 1.00 MAPT (0.42) MAPTALDH1A1LMNAHTTRAB9A
SCHEMBL463673 0.86 GRIN2D (0.52) MAPTALDH1A1LMNASMN1; SMN2GRIN2D
SCHEMBL3786399 0.83 PDE3B (0.50) MAPTALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL29909400 0.82 ALDH1A1 (0.47) MAPTALDH1A1LMNAHTTRAB9A
SCHEMBL30504341 0.82 KDM4E (0.47) MAPTALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL25201307 0.82 KDM4E (0.47) MAPTALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL2731858 0.82 ALDH1A1 (0.47) MAPTALDH1A1LMNAHTTRAB9A
SCHEMBL23172280 0.75 IDO1 (0.37) ALDH1A1SMN1; SMN2GRIN2DGRIN3BGRIN1
SCHEMBL16738736 0.73 EPAS1 (0.49) MAPTALDH1A1PDE3BPDE3AGRIN2D
SCHEMBL19644507 0.73 GRIA1 (0.50) MAPTALDH1A1LMNAHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022011274-A1 SUBSTITUTED 1,6-NAPHTHYRIDINE INHIBITORS OF CDK5 GOLDFINCH BIO, INC. (US) 2022-01-13 WO disclosed
WO-2020240492-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND THE PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2020-12-03 WO disclosed