SCHEMBL14403258

SCHEMBL14403258

Cc1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.65
ALDH1A1 P00352 2/20 0.65
KEAP1 Q14145 1/20 0.61
KMT2A Q03164 4/20 0.60
MEN1 O00255 3/20 0.60
MAPT P10636 3/20 0.60
LMNA P02545 2/20 0.60
HTT P42858 2/20 0.60
TSHR P16473 1/20 0.60
HDAC4 P56524 1/20 0.58
HDAC6 Q9UBN7 1/20 0.58
HSD11B1 P28845 1/20 0.56
SLC40A1 Q9NP59 1/20 0.56
UQCRB P14927 1/20 0.52
HSD17B2 P37059 1/20 0.52
GAA P10253 1/20 0.52
MCL1 Q07820 1/20 0.52
ACLY P53396 1/20 0.52
USP2 O75604 1/20 0.51
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7588697 0.89 PTGES2 (0.74) PTGES2KMT2AMEN1MAPTLMNA
SCHEMBL7589492 0.84 PTGES2 (0.56) PTGES2ALDH1A1KMT2AMEN1MAPT
SCHEMBL13875339 0.82 ALDH1A1 (0.71) ALDH1A1KEAP1KMT2AMEN1TSHR
SCHEMBL16325550 0.82 FFAR4 (0.63) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL13615288 0.82 HSD17B2 (0.57) PTGES2HSD11B1UQCRBHSD17B2CYP2C9
SCHEMBL4623054 0.82 ALDH1A1 (0.75) ALDH1A1KEAP1KMT2AMEN1MAPT
SCHEMBL834586 0.82 ALDH1A1 (0.75) ALDH1A1KEAP1KMT2AMEN1MAPT
SCHEMBL1116405 0.81 ALDH1A1 (0.74) ALDH1A1KEAP1KMT2AMEN1MAPT
SCHEMBL30102910 0.81 ALDH1A1 (0.74) ALDH1A1KEAP1KMT2AMEN1MAPT
SCHEMBL29540970 0.81 KEAP1 (0.68) PTGES2KEAP1KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007112998-A1 3-UNSUBSTITUTED N-(ARYL- OR HETEROARVL)-PYRAZOLORI [1,5-A]PYRIMIDINES AS KINASE INHIBITORS NOVARTIS AG (CH) 2007-10-11 WO disclosed