SCHEMBL14403274

SCHEMBL14403274

Cc1nc(C)c(-c2ccn(CCCCN3CC4CC4C3)c(=O)n2)s1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 4/20 0.34
CCNE1 P24864 2/20 0.34
CDK4 P11802 1/20 0.34
DRD2 P14416 8/20 0.34
DRD3 P35462 8/20 0.34
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
AURKA O14965 1/20 0.33
CDK9 P50750 1/20 0.33
AURKB Q96GD4 1/20 0.33
KDR P35968 1/20 0.32
COMT P21964 4/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
NPY5R Q15761 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568757 0.82 CDK2 (0.41) CDK2CCNE1CDK4AURKACDK9
SCHEMBL14401137 0.62 CDK4 (0.47) CDK2CCNE1CDK4AURKACDK9
SCHEMBL5717577 0.61 CDK4 (0.38) CDK2CCNE1CDK4COMTLMNA
SCHEMBL2353217 0.60 DRD2 (0.51) DRD2DRD3KDR
SCHEMBL2347681 0.59 TLR8 (0.43) DRD2DRD3KDR
SCHEMBL3572766 0.58 TGFBR1 (0.37) DRD2DRD3
SCHEMBL3574498 0.58 CCR1 (0.43) DRD2DRD3KDRLMNA
SCHEMBL3571130 0.58 TLR8 (0.46) LMNA
SCHEMBL3572286 0.57 CDK2 (0.49) CDK2CCNE1CDK4AURKACDK9
SCHEMBL2351423 0.57 TLR8 (0.44) CDK4DRD2DRD3KDRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007113260-A1 AZABICYCLO [3. 1. O] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2007-10-11 WO disclosed