SCHEMBL14404689

SCHEMBL14404689

CN1CCCC1CCn1c(Cc2ccc(OI)cc2)cc2cc(NC(=N)c3cccs3)ccc21

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 15/20 0.52
NOS1 P29475 15/20 0.52
OPRM1 P35372 2/20 0.46
NOS2 P35228 9/20 0.40
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2262457 0.91 NOS3 (0.51) NOS3NOS1OPRM1NOS2
SCHEMBL12391672 0.91 NOS3 (0.54) NOS3NOS1OPRM1NOS2KCNH2
SCHEMBL2262112 0.91 NOS3 (0.62) NOS3NOS1OPRM1NOS2KCNH2
SCHEMBL1122087 0.84 NOS3 (0.69) NOS3NOS1OPRM1NOS2KCNH2
SCHEMBL2263080 0.82 NOS3 (0.49) NOS3NOS1OPRM1NOS2KCNH2
SCHEMBL14388882 0.80 NOS3 (0.46) NOS3NOS1OPRM1NOS2KCNH2
SCHEMBL1593998 0.79 OPRM1 (0.71) NOS3NOS1OPRM1NOS2
SCHEMBL14618254 0.78 OPRM1 (0.62) NOS3NOS1OPRM1NOS2
SCHEMBL15178523 0.77 NOS3 (0.36) NOS3NOS1OPRM1
SCHEMBL12367461 0.77 SMN1; SMN2 (0.38) NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007118314-A1 1,5 AND 3,6- SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2007-10-25 WO disclosed