SCHEMBL14409016

SCHEMBL14409016

CC(C)Cc1cnc(-c2ccccc2)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.52
CYP11B2 P19099 2/20 0.52
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 1/20 0.45
LMNA P02545 6/20 0.45
ALDH1A1 P00352 7/20 0.43
SMN1; SMN2 Q16637 6/20 0.43
NPC1 O15118 6/20 0.43
RAB9A P51151 6/20 0.43
KDM4E B2RXH2 3/20 0.43
NFKB1 P19838 3/20 0.43
NFKB2 Q00653 3/20 0.43
RELA Q04206 3/20 0.43
HPGDS O60760 2/20 0.43
MAPT P10636 4/20 0.41
HPGD P15428 2/20 0.41
QPCT Q16769 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
FBP1 P09467 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16402703 0.83 SMN1; SMN2 (0.44) CYP11B1CYP11B2LMNAALDH1A1SMN1; SMN2
SCHEMBL153089 0.80 CYP11B1 (0.56) CYP11B1CYP11B2HDAC1HDAC2LMNA
SCHEMBL13437308 0.79 ALDH1A1 (0.50) LMNAALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL12890736 0.79 CYP11B1 (0.49) CYP11B1CYP11B2HDAC1HDAC2LMNA
SCHEMBL2095827 0.78 CYP11B1 (0.54) CYP11B1CYP11B2HDAC1HDAC2LMNA
SCHEMBL28296261 0.78 CYP11B1 (0.41) CYP11B1CYP11B2LMNAALDH1A1SMN1; SMN2
SCHEMBL20011457 0.78 CYP11B1 (0.55) CYP11B1CYP11B2HDAC1HDAC2LMNA
SCHEMBL12844399 0.77 CYP11B1 (0.54) CYP11B1CYP11B2HDAC1HDAC2LMNA
SCHEMBL2226354 0.77 CYP11B1 (0.53) CYP11B1CYP11B2HDAC1HDAC2LMNA
SCHEMBL6973608 0.77 CYP11B1 (0.53) CYP11B1CYP11B2HDAC1HDAC2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7273876-B2 Substituted bicylic thiophene derivatives, compositions containing such compounds and methods of use MERCK & CO., INC. (US) 2007-09-25 US disclosed