SCHEMBL14409802

SCHEMBL14409802

CC(=O)N(I)c1ccc(-c2c(C#N)c(N)nc(Sc3ccccc3)c2C#N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.51
NPSR1 Q6W5P4 3/20 0.51
RXFP1 Q9HBX9 2/20 0.51
ADORA1 P30542 7/20 0.48
ADORA2B P29275 2/20 0.48
ADORA2A P29274 2/20 0.48
ADORA3 P0DMS8 1/20 0.48
KDM4E B2RXH2 5/20 0.46
HSD17B10 Q99714 5/20 0.46
ALOX15 P16050 4/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPK1 P28482 2/20 0.46
HTT P42858 2/20 0.46
LMNA P02545 1/20 0.46
ABL1 P00519 1/20 0.45
RET P07949 1/20 0.45
ALK Q9UM73 1/20 0.45
ALDH1A1 P00352 6/20 0.45
HPGD P15428 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3556602 0.83 ADORA2B (0.68) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL245593 0.81 ADORA1 (0.64) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL13938147 0.80 ADORA1 (0.62) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL244863 0.78 ADORA1 (0.61) MAPTNPSR1RXFP1ADORA1ADORA2A
SCHEMBL3333404 0.77 MAPT (0.81) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL15286658 0.75 ADORA1 (0.64) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL4034485 0.74 MAPT (0.63) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL28185531 0.74 KDM4E (0.73) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL241556 0.74 MAPT (0.59) MAPTNPSR1RXFP1ADORA1ADORA2B
SCHEMBL6462984 0.74 MAPT (0.59) MAPTNPSR1RXFP1ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1417173-B1 SUBSTITUTED 2-THIO-3, 5-DICYANO-4-PHENYL-6-AMINOPYRIDINES AND THEIR USE AS ADENOSINE RECEPTOR-SELECTIVE LIGANDS BAYER HEALTHCARE AG (DE) 2007-09-26 EP disclosed