SCHEMBL1441295

SCHEMBL1441295

NC(=O)c1c(O)c2ccccc2n(C2CC2)c1=O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.66
KMT2A Q03164 4/20 0.66
ALDH1A1 P00352 3/20 0.66
PADI4 Q9UM07 1/20 0.44
OPRM1 P35372 2/20 0.44
OPRD1 P41143 2/20 0.44
OPRK1 P41145 2/20 0.44
OGFRL1 Q5TC84 2/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
GAA P10253 1/20 0.43
PPARG P37231 1/20 0.43
NCOA2 Q15596 1/20 0.43
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
POLB P06746 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1441135 0.94 MEN1 (0.74) MEN1KMT2AALDH1A1PADI4OPRM1
SCHEMBL1440437 0.93 MEN1 (0.77) MEN1KMT2AALDH1A1OPRM1OPRD1
SCHEMBL11372663 0.82 ALDH1A1 (0.76) MEN1KMT2AALDH1A1PADI4OPRM1
SCHEMBL31423075 0.80 ALDH1A1 (0.56) MEN1KMT2AALDH1A1PADI4OPRM1
SCHEMBL28859816 0.76 MEN1 (0.46) MEN1KMT2AALDH1A1PADI4OPRM1
SCHEMBL35212365 0.76 ALDH1A1 (0.74) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL10962357 0.76 ALDH1A1 (0.74) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL10680267 0.76 MEN1 (0.60) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL11377355 0.75 ALDH1A1 (0.69) MEN1KMT2AALDH1A1OPRM1OPRD1
SCHEMBL5332461 0.74 ALDH1A1 (0.71) MEN1KMT2AALDH1A1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2507225-A1 L -DIHYDRO-2-OXOQUINOLINE COMPOUNDS A 5-HT4 RECEPTOR LIGANDS Suven Life Sciences Limited (IN) 2012-10-10 EP claimed
WO-2011030349-A1 L -DIHYDRO-2-OXOQUINOLINE COMPOUNDS A 5-HT4 RECEPTOR LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2011-03-17 WO claimed
EP-2507225-A1 L -DIHYDRO-2-OXOQUINOLINE COMPOUNDS A 5-HT4 RECEPTOR LIGANDS Suven Life Sciences Limited (IN) 2012-10-10 EP disclosed