SCHEMBL14419600

SCHEMBL14419600

CC(=O)Nc1ccc(S(=O)(=O)NCC2CC2)cc1C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.61
PDK1 Q15118 1/20 0.54
PDK2 Q15119 1/20 0.54
PDK3 Q15120 1/20 0.54
PDK4 Q16654 1/20 0.54
PPARG P37231 1/20 0.53
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
ALDH1A1 P00352 3/20 0.53
CYP2C9 P11712 1/20 0.53
HPGD P15428 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
LMNA P02545 2/20 0.50
TP53 P04637 1/20 0.50
BACE1 P56817 1/20 0.50
POLB P06746 1/20 0.50
THRB P10828 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
PARG Q86W56 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14419684 0.83 POLB (0.64) MEN1KMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL14419466 0.82 BACE1 (0.55) CCR8PPARGALDH1A1HPGDSMN1; SMN2
SCHEMBL14419634 0.80 PPARG (0.53) PDK1PDK2PDK3PDK4PPARG
SCHEMBL14419470 0.80 ALDH1A1 (0.57) PPARGMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL14419631 0.78 RAB9A (0.68) KMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL14419602 0.77 PARG (0.55) CCR8MEN1KMT2AALDH1A1CYP2C9
SCHEMBL24997782 0.76 CCR8 (1.00) CCR8
SCHEMBL4397776 0.76 MEN1 (0.68) MEN1KMT2AALDH1A1CYP2C9HPGD
SCHEMBL4397778 0.76 MEN1 (0.68) MEN1KMT2AALDH1A1CYP2C9HPGD
SCHEMBL14419664 0.76 ALDH1A1 (0.60) KMT2AALDH1A1SMN1; SMN2LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7273863-B1 Benzophenones as inhibitors of reverse transcriptase SMITHKLINE BEECHAM CORPORATION (US) 2007-09-25 US disclosed