SCHEMBL14435398

SCHEMBL14435398

O=C(N[SH](=O)=O)c1ccc2c(C3CCCCC3)c3n(c2c1)CCNc1ccccc1-3

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.48
NR1I2 O75469 5/20 0.42
PRKCA P17252 1/20 0.40
MMP12 P39900 1/20 0.40
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
KCNH2 Q12809 2/20 0.35
SCN5A Q14524 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL804196 0.87 PRKCA (0.51) SCN9ANR1I2PRKCAMMP12CYP3A4
SCHEMBL14253483 0.86 SCN9A (0.55) SCN9ANR1I2PRKCAMMP12KCNH2
SCHEMBL14253482 0.86 SCN9A (0.67) SCN9ANR1I2KCNH2SCN5A
SCHEMBL4825561 0.85 SCN9A (0.45) SCN9ANR1I2PRKCAMMP12CYP3A4
SCHEMBL14435944 0.85 SCN9A (0.43) SCN9ANR1I2PRKCAMMP12KCNH2
SCHEMBL14253464 0.84 NR1I2 (0.60) SCN9ANR1I2PRKCAMMP12CYP3A4
SCHEMBL14435969 0.83 SCN9A (0.47) SCN9ANR1I2PRKCAMMP12CYP3A4
SCHEMBL14435393 0.82 SCN9A (0.46) SCN9ANR1I2PRKCAMMP12CYP3A4
SCHEMBL14253186 0.81 PRKCA (0.49) SCN9ANR1I2PRKCAMMP12CYP3A4
SCHEMBL3577991 0.81 SCN9A (0.47) SCN9ANR1I2PRKCAMMP12KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007092000-A1 INHIBITORS OF HCV REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-16 WO disclosed