SCHEMBL14435440

SCHEMBL14435440

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C(C(=O)O)CNc1ccccc1-3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.39
MMP12 P39900 1/20 0.39
SCN9A Q15858 6/20 0.38
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
ALDH1A1 P00352 4/20 0.36
NPSR1 Q6W5P4 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ATM Q13315 1/20 0.36
CYP3A4 P08684 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP2C9 P11712 2/20 0.35
NR1I2 O75469 2/20 0.35
CYP2D6 P10635 1/20 0.35
CNR2 P34972 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
CCNB2 O95067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14435438 0.89 PRKCA (0.37) PRKCAMMP12SCN9ABRD4CREBBP
SCHEMBL14253899 0.87 NR1I2 (0.44) PRKCAMMP12SCN9ABRD4CREBBP
SCHEMBL14253893 0.84 PRKCA (0.40) PRKCAMMP12SCN9AALDH1A1NPSR1
SCHEMBL14253454 0.83 PRKCA (0.46) PRKCAMMP12SCN9ABRD4CREBBP
SCHEMBL3574582 0.82 PRKCA (0.44) PRKCAMMP12SCN9ABRD4CREBBP
SCHEMBL4825561 0.82 SCN9A (0.45) PRKCAMMP12SCN9ABRD4CREBBP
SCHEMBL3577991 0.81 SCN9A (0.47) PRKCAMMP12SCN9ABRD4CREBBP
SCHEMBL13841666 0.79 ALDH1A1 (0.43) PRKCAMMP12SCN9AALDH1A1NPSR1
SCHEMBL3242888 0.79 ALDH1A1 (0.43) PRKCAMMP12SCN9AALDH1A1NPSR1
SCHEMBL804192 0.78 PRKCA (0.44) PRKCAMMP12SCN9ACYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007092000-A1 INHIBITORS OF HCV REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-16 WO disclosed