Erufosine

Erufosine

SCHEMBL14447882

CCCCCCCC/C=C\CCCCCCCCCCCCOP(=O)(O)OCC[N+](C)(C)C

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LPAR3 Q9UBY5 6/20 0.60
LPAR2 Q9HBW0 5/20 0.60
LPAR1 Q92633 3/20 0.60
LMNA P02545 1/20 0.59
ESR1 P03372 1/20 0.59
ADORA3 P0DMS8 1/20 0.59
CDC25A P30304 1/20 0.59
AGTR1 P30556 1/20 0.59
AKT1 P31749 1/20 0.59
ADRA1A P35348 1/20 0.59
KCNH2 Q12809 1/20 0.59
P2RY10 O00398 5/20 0.54
MEN1 O00255 1/20 0.51
S1PR1 P21453 1/20 0.51
KMT2A Q03164 1/20 0.51
FABP3 P05413 1/20 0.50
GPR34 Q9UPC5 1/20 0.50
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14448106 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
Erufosine SCHEMBL52781 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
SCHEMBL7068514 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
SCHEMBL17817094 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
SCHEMBL17817487 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
SCHEMBL9027644 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
Erufosine SCHEMBL14448104 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
Elaidylphosphocholine SCHEMBL12235518 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
Elaidylphosphocholine SCHEMBL515227 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1
SCHEMBL14447795 1.00 LPAR3 (0.60) LPAR3LPAR2LPAR1LMNAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240238253-A1 SPRAY-DRIED DISPERSIONS, FORMULATIONS, AND POLYMORPHS OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TRIFLUOROPROPAN-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE LOXO ONCOLOGY, INC. 2024-07-18 US disclosed
WO-2024112654-A1 SPIROCYCLIC DIHYDROPYRANOPYRIMIDINE KRAS INHIBITORS Treeline Biosciences, Inc. (US) 2024-05-30 WO disclosed
US-20240158376-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. 2024-05-16 US disclosed
WO-2024097636-A1 COMBINATION THERAPY FOR TREATING CANCER SCORPION THERAPEUTICS, INC. (US) 2024-05-10 WO disclosed
EP-4363414-A1 COMPOUNDS THAT INHIBIT PI3K ISOFORM ALPHA AND METHODS FOR TREATING CANCER Scorpion Therapeutics, Inc. (US) 2024-05-08 EP disclosed
WO-2024086804-A1 INDOLIZINE DERIVATIVES FOR TREATING CANCER SCORPION THERAPEUTICS, INC. (US) 2024-04-25 WO disclosed
WO-2024086809-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. (US) 2024-04-25 WO disclosed
US-11965178-B2 Platelets loaded with anti-cancer agents CELLPHIRE, INC. (US) 2024-04-23 US disclosed
WO-2024077036-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. (US) 2024-04-11 WO disclosed
EP-4346815-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Schrödinger, Inc. (US) 2024-04-10 EP disclosed
US-20200087399-A1 PHOSPHOLIPID ETHER (PLE) CAR T CELL TUMOR TARGETING (CTCT) AGENTS Seattle Children's Hospital (dba Seattle Children's Research Institute) 2020-03-19 US disclosed
WO-2020033272-A1 METHODS AND COMPOSITIONS FOR STIMULATION OF CHIMERIC ANTIGEN RECEPTOR T CELLS WITH HAPTEN LABELLED CELLS Seattle Children's Hospital (dba Seattle Children's Research Institute) (US) 2020-02-13 WO disclosed
WO-2020028258-A1 SPRAY-DRIED DISPERSIONS AND FORMULATIONS OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TRIFLUORO PROPAN-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE LOXO ONCOLOGY, INC. (US) 2020-02-06 WO disclosed
WO-2019191659-A1 TREATMENT OF TRK-ASSOCIATED CANCERS LOXO ONCOLOGY, INC. (US) 2019-10-03 WO disclosed
US-20190256924-A1 METHODS AND MATERIALS FOR ASSESSING AND TREATING CANCER THE JOHNS HOPKINS UNIVERSITY 2019-08-22 US disclosed
WO-2019156795-A1 FLUORESCEIN-SPECIFIC CARS EXHIBITING OPTIMAL T CELL FUNCTION AGAINST FL-PLE LABELLED TUMORS Seattle Children's Hospital (dba Seattle Children's Research Institute) (US) 2019-08-15 WO disclosed
WO-2019067092-A1 METHODS AND MATERIALS FOR ASSESSING AND TREATING CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2019-04-04 WO disclosed
WO-2018148224-A1 PHOSPHOLIPID ETHER (PLE) CAR T CELL TUMOR TARGETING (CTCT) AGENTS Seattle Children's Hospital (dba Seattle Children's Research Institute) (US) 2018-08-16 WO disclosed
US-20070167408-A1 NOVEL ALKYL PHOSPHOLIPID DERIVATIVES WITH REDUCED CYTOTOXICITY AND USES THEREOF ZENTARIS GMBH (DE) 2007-07-19 US disclosed
EP-1800684-A1 Novel alkyl phospholipid derivatives and uses thereof Zentaris GmbH (DE) 2007-06-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240158376-A1 METHODS FOR TREATING CANCER PIK3CA, PTEN, BRCA1 LPAR3 687/4885LPAR2 603/4885LPAR1 917/4885
US-20070167408-A1 NOVEL ALKYL PHOSPHOLIPID DERIVATIVES WITH REDUCED CYTOTOXICITY AND USES THEREOF PHOSPHO1, PTDSS1, PTDSS2 LPAR3 82/4885LPAR2 88/4885LPAR1 74/4885
US-20240238253-A1 SPRAY-DRIED DISPERSIONS, FORMULATIONS, AND POLYMORPHS OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TRIFLUOROPROPAN-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE API5, IL5, SRMS LPAR3 2762/4885LPAR2 3377/4885LPAR1 3624/4885
US-20200087399-A1 PHOSPHOLIPID ETHER (PLE) CAR T CELL TUMOR TARGETING (CTCT) AGENTS PHOSPHO1, LCAT, CD47 LPAR3 84/4885LPAR2 67/4885LPAR1 49/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.