SCHEMBL1445168

SCHEMBL1445168

NC(=O)c1cccc(-c2ccncn2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.52
KDM1A O60341 1/20 0.50
HPGDS O60760 1/20 0.49
PIM1 P11309 1/20 0.48
PRKCI P41743 1/20 0.48
CCNT1 O60563 1/20 0.46
CCND1 P24385 1/20 0.46
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
CDK7 P50613 1/20 0.46
CDK9 P50750 1/20 0.46
CCNH P51946 1/20 0.46
MNAT1 P51948 1/20 0.46
CDK6 Q00534 1/20 0.46
PARP1 P09874 5/20 0.44
CSNK2A2 P19784 2/20 0.44
CSNK2B P67870 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ABL1 P00519 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30285920 0.85 KMO (0.57) KDM4EABL1BCRGRM5
SCHEMBL940865 0.85 KMO (0.57) KDM4EABL1BCRGRM5
SCHEMBL7824311 0.84 ASIC3 (0.43) FYNHPGDSMAPK1GRM5GSK3B
Hydrochloric Acid SCHEMBL7816742 0.83 ASIC3 (0.43) FYNMAPK1GRM5GSK3B
SCHEMBL29818231 0.82 ROCK1 (0.49) KDM4EABL1MAPTBCRMAPK1
SCHEMBL8706110 0.82 ROCK1 (0.41) FYNMAPK1GRM5GSK3BSIRT2
SCHEMBL167080 0.81 CHEK2 (0.57) FYNKDM1AHPGDSPIM1PRKCI
SCHEMBL18209898 0.81 CCNT1 (0.49) FYNKDM1AHPGDSPIM1PRKCI
SCHEMBL1445286 0.81 MAP4K4 (0.54) FYNMAPK1GSK3B
SCHEMBL30036208 0.81 CHEK2 (0.57) FYNKDM1AHPGDSPIM1PRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2480235-A2 NOVEL IODO PYRIMIDINE DERIVATIVES USEFUL FOR THE TREATMENT OF MACROPHAGE MIGRATION INHIBITORY FACTOR (MIF)-IMPLICATED DISEASES AND CONDITIONS University Of Louisville Research Foundation, Inc. (US) 2012-08-01 EP claimed
WO-2011038234-A2 NOVEL IODO PYRIMIDINE DERIVATIVES USEFUL FOR THE TREATMENT OF MACROPHAGE MIGRATION INHIBITORY FACTOR (MIF)-IMPLICATED DISEASES AND CONDITIONS UNIVERSITY OF LOUISVILLE RESEARCH FOUNDATION, INC. (US) 2011-03-31 WO claimed