SCHEMBL14463582

SCHEMBL14463582

CCOc1ccc(-n2c(NCc3ccc(C(C)(C)C)cc3)nc3ccc(CI)cc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
EPHX2 P34913 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
GAA P10253 3/20 0.42
ALDH1A1 P00352 4/20 0.42
TP53 P04637 4/20 0.42
MAPT P10636 5/20 0.41
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 1/20 0.41
CACNA2D1 P54289 4/20 0.40
HPGD P15428 1/20 0.39
LMNA P02545 1/20 0.39
CNR2 P34972 1/20 0.38
MEN1 O00255 1/20 0.38
APP P05067 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
MAPK1 P28482 1/20 0.38
SNCA P37840 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14463835 0.93 NPC1 (0.41) NPC1RAB9AEPHX2NR1H4GAA
SCHEMBL14463585 0.93 NPC1 (0.41) NPC1RAB9AEPHX2NR1H4GAA
SCHEMBL14463414 0.92 NPC1 (0.47) NPC1RAB9AEPHX2NR1H4GAA
SCHEMBL14463903 0.92 NPC1 (0.56) NPC1RAB9AGAAALDH1A1TP53
SCHEMBL14463475 0.90 NPC1 (0.39) NPC1RAB9AEPHX2NR1H4GAA
SCHEMBL14463444 0.90 NPC1 (0.47) NPC1RAB9AEPHX2NR1H4GAA
SCHEMBL4930629 0.89 NPC1 (0.50) NPC1RAB9AEPHX2NR1H4GAA
SCHEMBL14463413 0.88 NPC1 (0.52) NPC1RAB9AGAAALDH1A1TP53
SCHEMBL14463583 0.88 EPHX2 (0.43) NPC1RAB9AEPHX2NR1H4TP53
Hydrochloric Acid SCHEMBL4932676 0.88 NPC1 (0.49) NPC1RAB9AEPHX2NR1H4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1810677-A1 RECEPTOR FUNCTION REGULATING AGENT Takeda Pharmaceutical Company Limited (JP) 2007-07-25 EP disclosed