SCHEMBL14463583

SCHEMBL14463583

CC(C)(C)c1ccc(CNc2nc3ccc(CI)cc3n2-c2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
TRPC5 Q9UL62 1/20 0.41
TRPV1 Q8NER1 2/20 0.37
KCNN3 Q9UGI6 1/20 0.37
PPARG P37231 2/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PPARA Q07869 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CACNA1H O95180 1/20 0.35
P2RX7 Q99572 1/20 0.35
GPR39 O43194 1/20 0.35
CYP3A4 P08684 1/20 0.35
BRD4 O60885 1/20 0.35
NTRK1 P04629 1/20 0.35
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14463870 0.92 TRPV1 (0.40) EPHX2NR1H4TRPC5TRPV1KCNN3
SCHEMBL14463910 0.90 EPHX2 (0.42) EPHX2NR1H4TRPC5TRPV1KCNN3
SCHEMBL14463475 0.89 NPC1 (0.39) EPHX2NR1H4NPC1RAB9ALMNA
SCHEMBL4931809 0.89 CYP3A4 (0.44) EPHX2NR1H4TRPC5TRPV1KCNN3
SCHEMBL14463582 0.88 NPC1 (0.50) EPHX2NR1H4L3MBTL1NPC1RAB9A
SCHEMBL14463835 0.86 NPC1 (0.41) EPHX2NR1H4POLBNPC1RAB9A
SCHEMBL14463585 0.86 NPC1 (0.41) EPHX2NR1H4L3MBTL1NPC1RAB9A
SCHEMBL4922605 0.86 TRPC5 (0.45) EPHX2NR1H4TRPC5TRPV1KCNN3
SCHEMBL14463473 0.81 TRPC5 (0.37) TRPC5NPC1RAB9ATP53CYP3A4
SCHEMBL4927317 0.81 P2RX3 (0.41) EPHX2NR1H4TRPC5TRPV1KCNN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1810677-A1 RECEPTOR FUNCTION REGULATING AGENT Takeda Pharmaceutical Company Limited (JP) 2007-07-25 EP disclosed