SCHEMBL14465248

SCHEMBL14465248

CCOC(=O)NCCNc1ccnc(-c2c[nH]c3ncc(Cl)cc23)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.44
CYP3A4 P08684 5/20 0.44
ALDH1A1 P00352 4/20 0.44
CLK4 Q9HAZ1 4/20 0.44
HSD17B10 Q99714 2/20 0.44
MAPK1 P28482 2/20 0.44
ALOX15 P16050 2/20 0.44
JAK2 O60674 2/20 0.40
ROCK2 O75116 2/20 0.40
CDK9 P50750 2/20 0.40
PLK4 O00444 1/20 0.40
STK10 O94804 1/20 0.40
ABL1 P00519 1/20 0.40
PRKCB P05771 1/20 0.40
MET P08581 1/20 0.40
TOP2A P11388 1/20 0.40
PRKCA P17252 1/20 0.40
CSNK2A2 P19784 1/20 0.40
JAK1 P23458 1/20 0.40
MARK3 P27448 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14465240 0.90 ALDH1A1 (0.40) CYP1A2CYP3A4ALDH1A1CLK4HSD17B10
SCHEMBL14465256 0.83 ALDH1A1 (0.40) CYP1A2CYP3A4ALDH1A1CLK4HSD17B10
SCHEMBL14327614 0.81 CLK4 (0.46) CYP1A2CYP3A4ALDH1A1CLK4MAPK1
SCHEMBL14712339 0.81 JAK2 (0.49) CYP1A2CYP3A4ALDH1A1CLK4MAPK1
SCHEMBL24059738 0.78 CYP1A2 (0.38) CYP1A2CYP3A4ALDH1A1CLK4MAPK1
SCHEMBL2630217 0.77 JAK3 (0.48) CLK4JAK2ROCK2CDK9PLK4
SCHEMBL2630148 0.77 JAK3 (0.49) CYP3A4JAK2ROCK2CDK9PLK4
SCHEMBL15723264 0.76 CCNT1 (0.42) CDK9JAK3
SCHEMBL10303502 0.76 CCNT1 (0.42) CDK9JAK3
SCHEMBL2633664 0.76 JAK2 (0.52) CYP1A2CYP3A4ALDH1A1JAK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007084557-A2 AZAINDOLES USEFUL AS INHIBITORS OF JANUS KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-07-26 WO disclosed