SCHEMBL1447151

SCHEMBL1447151

O=C(c1ccc(Br)cc1F)N1CCCOCC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
TSHR P16473 1/20 0.52
EPHX2 P34913 2/20 0.52
SLC6A5 Q9Y345 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 4/20 0.48
MEN1 O00255 1/20 0.48
CNR1 P21554 3/20 0.48
CPS1 P31327 1/20 0.48
CCKBR P32239 1/20 0.46
GAA P10253 1/20 0.46
ERN1 O75460 1/20 0.46
DGAT1 O75907 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29897652 0.94 MAPT (0.57) MAPTTSHREPHX2SLC6A5RAB9A
SCHEMBL968813 0.94 MAPT (0.57) MAPTTSHREPHX2SLC6A5RAB9A
SCHEMBL643698 0.87 CPS1 (0.60) MAPTRAB9AKMT2ACPS1CCKBR
SCHEMBL1424241 0.87 CCKBR (0.56) MAPTTSHRRAB9AKMT2ACNR1
SCHEMBL30791513 0.87 CCKBR (0.56) MAPTTSHRRAB9AKMT2ACNR1
SCHEMBL969401 0.86 CCKBR (0.58) MAPTTSHRRAB9AKMT2AMEN1
SCHEMBL1447765 0.84 MAPT (0.56) MAPTTSHRRAB9AKMT2ACNR1
SCHEMBL17400734 0.84 MAPT (0.52) MAPTTSHREPHX2KMT2AMEN1
SCHEMBL1447782 0.84 HPGD (0.50) MAPTSLC6A5RAB9AKMT2AMEN1
SCHEMBL16379735 0.83 MAPT (0.57) MAPTTSHREPHX2SLC6A5RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2301928-A1 Imidazolyl-pyrimidine compounds for use in the treatment of proliferative disorders AstraZeneca AB (SE) 2011-03-30 EP disclosed
US-20080280906-A1 Imidazolyl-Pyrimidine Compounds for Use in the Treatment of Proliferative Disorders ASTRAZENECA AB (SE) 2008-11-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280906-A1 Imidazolyl-Pyrimidine Compounds for Use in the Treatment of Proliferative Disorders CCNI, MKI67, TYMP MAPT 3364/4885TSHR 3665/4885EPHX2 2669/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.