SCHEMBL14498121

SCHEMBL14498121

N#C/N=C1\Nc2ccccc2CN1C1CCNCC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.41
HTR2A P28223 5/20 0.41
HTR2B P41595 4/20 0.39
PARP1 P09874 2/20 0.37
CALCRL Q16602 2/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
TNKS O95271 1/20 0.32
HTR5A P47898 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CTSS P25774 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11097882 0.99 HTR2C (0.40) HTR2CHTR2AHTR2BPARP1CALCRL
Hydrochloric Acid SCHEMBL11160630 0.99 HTR2C (0.40) HTR2CHTR2AHTR2BPARP1CALCRL
SCHEMBL5369548 0.87 BRD4 (0.33) CALCRLBRD4CREBBPTNKSHTR5A
SCHEMBL14410233 0.82 PARP1 (0.40) PARP1CALCRLBRD4CREBBPCTSS
SCHEMBL11102413 0.78 MAPK1 (0.48) CALCRL
SCHEMBL11102417 0.78 MAPK1 (0.48) CALCRL
SCHEMBL31184539 0.76 BRD4 (0.50) HTR2CHTR2AHTR2BPARP1CALCRL
SCHEMBL2100919 0.76 BRD4 (0.50) HTR2CHTR2AHTR2BPARP1CALCRL
SCHEMBL31184549 0.76 BRD4 (0.50) HTR2CHTR2AHTR2BPARP1CALCRL
SCHEMBL14417234 0.75 HTR2C (0.43) HTR2CHTR2AHTR2BPARP1CALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7230001-B1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2007-06-12 US disclosed