SCHEMBL5369548

SCHEMBL5369548

N#CN=C1Nc2ccccc2CN1C1CC[N]CC1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
CTSS P25774 9/20 0.32
HTR5A P47898 3/20 0.32
CALCRL Q16602 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TNKS O95271 1/20 0.31
PTK2B Q14289 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14498121 0.87 HTR2C (0.41) BRD4CREBBPCTSSHTR5ACALCRL
Hydrochloric Acid SCHEMBL11160630 0.86 HTR2C (0.40) BRD4CREBBPHTR5ACALCRLALDH1A1
Hydrochloric Acid SCHEMBL11097882 0.86 HTR2C (0.40) BRD4CREBBPHTR5ACALCRLALDH1A1
SCHEMBL14410233 0.82 PARP1 (0.40) BRD4CREBBPCTSSCALCRL
SCHEMBL3279615 0.76 BRD4 (0.50) BRD4CREBBPCTSSCALCRL
SCHEMBL11102413 0.76 MAPK1 (0.48) CALCRL
SCHEMBL11102417 0.76 MAPK1 (0.48) CALCRL
SCHEMBL5374765 0.75 QPCT (0.40) BRD4CREBBPCTSSHTR5ACALCRL
SCHEMBL5377735 0.70 OPRM1 (0.49) CTSSCALCRL
SCHEMBL11100446 0.70 KCNH2 (0.33) CALCRLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070208036-A1 Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and processes for preparing them BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2007-09-06 US claimed
US-20070208036-A1 Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and processes for preparing them BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2007-09-06 US disclosed
US-7230001-B1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2007-06-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070208036-A1 Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and processes for preparing them ARRB1, NPY1R, ADRB3 BRD4 3076/4885CREBBP 2215/4885CTSS 558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.