SCHEMBL14498481

SCHEMBL14498481

C=CC[C@]1(C)CCCCC1=O

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.32
POLB P06746 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
LMNA P02545 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23463949 1.00 CYP19A1 (0.32) CYP19A1POLBMEN1KMT2AALDH1A1
SCHEMBL1137957 1.00 CYP19A1 (0.32) CYP19A1POLBMEN1KMT2AALDH1A1
SCHEMBL14498509 0.98 POLB (0.34) CYP19A1POLBMEN1KMT2AALDH1A1
SCHEMBL14498540 0.98 POLB (0.34) CYP19A1POLBMEN1KMT2AALDH1A1
SCHEMBL18093583 0.98 POLB (0.34) CYP19A1POLBMEN1KMT2AALDH1A1
SCHEMBL23687486 0.94 CYP19A1 (0.33) CYP19A1
SCHEMBL11725794 0.94 CYP19A1 (0.33) CYP19A1
SCHEMBL23687485 0.94 CYP19A1 (0.33) CYP19A1
Acetic Acid SCHEMBL8453705 0.92 MEN1 (0.40) POLBMEN1KMT2AALDH1A1
SCHEMBL31268499 0.82 POLB (0.33) CYP19A1POLBGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250391519-A1 CHEMICAL SYNTHESIS PLATFORM UNIV GLASGOW COURT (GB) 2025-12-25 US disclosed
EP-4548355-A1 CHEMICAL SYNTHESIS PLATFORM The University Court Of The University Of Glasgow (GB) 2025-05-07 EP disclosed
WO-2024003151-A1 CHEMICAL SYNTHESIS PLATFORM THE UNIVERSITY COURT OF THE UNIVERSITY OF GLASGOW (GB) 2024-01-04 WO disclosed
EP-3274342-B1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INST OF TECHN (US) 2022-05-04 EP disclosed
EP-3274342-B1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INST OF TECHN (US) 2022-05-04 EP disclosed
US-20190055182-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY 2019-02-21 US disclosed
US-20190055182-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY 2019-02-21 US disclosed
US-10106479-B2 Asymmetric catalytic decarboxylative alkyl alkylation using low catalyst concentrations and a robust precatalyst CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-10-23 US disclosed
EP-3274342-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST California Institute of Technology (US) 2018-01-31 EP disclosed
WO-2016160579-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST STOLTZ BRIAN M (US) 2016-10-06 WO disclosed
WO-2016160579-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST STOLTZ BRIAN M (US) 2016-10-06 WO disclosed
US-20160280623-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY 2016-09-29 US disclosed
US-20160280623-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY 2016-09-29 US disclosed
US-20160280623-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY 2016-09-29 US disclosed
US-7235698-B2 Enantioselective, catalytic allylation of ketones and olefins CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2007-06-26 US disclosed
US-7235698-B2 Enantioselective, catalytic allylation of ketones and olefins CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2007-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160280623-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST IDH3B, IDH3A, CYP51A1 CYP19A1 30/4885POLB 274/4885MEN1 1312/4885
US-10106479-B2 Asymmetric catalytic decarboxylative alkyl alkylation using low catalyst concentrations and a robust precatalyst IDH3B, IDH3A, CYP51A1 CYP19A1 30/4885POLB 274/4885MEN1 1312/4885
US-20250391519-A1 CHEMICAL SYNTHESIS PLATFORM SET, CBS, COASY CYP19A1 218/4885POLB 1914/4885MEN1 820/4885
US-20190055182-A1 ASYMMETRIC CATALYTIC DECARBOXYLATIVE ALKYL ALKYLATION USING LOW CATALYST CONCENTRATIONS AND A ROBUST PRECATALYST IDH3B, IDH3A, CYP51A1 CYP19A1 30/4885POLB 274/4885MEN1 1312/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.