SCHEMBL14531996

SCHEMBL14531996

CC(=O)c1cccc(C(C#N)(C#N)C#N)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.37
CTSS P25774 3/20 0.37
P2RX7 Q99572 9/20 0.36
CTSK P43235 2/20 0.35
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.33
TAS1R3 Q7RTX0 2/20 0.33
TAS1R1 Q7RTX1 2/20 0.33
TAS1R2 Q8TE23 2/20 0.33
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
TAS2R14 Q9NYV8 1/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18511684 0.79 CA2 (0.43) PDK2CTSSP2RX7CTSKTSHR
SCHEMBL9524633 0.77 CTSS (0.56) CTSSP2RX7CTSKTAS2R14
SCHEMBL30562236 0.77 CTSS (0.56) CTSSP2RX7CTSKTAS2R14
SCHEMBL3781319 0.75 TSHR (0.48) PDK2TSHRTAS1R3TAS1R1TAS1R2
SCHEMBL8681119 0.74 NOTUM (0.41) TSHRHTTPOLBRAB9ASMN1; SMN2
SCHEMBL28659549 0.72 CTSS (0.42) PDK2CTSSP2RX7CTSKTAS2R14
SCHEMBL825860 0.72 TSHR (0.49) PDK2CTSSP2RX7CTSKTSHR
SCHEMBL826478 0.72 CTSS (0.36) PDK2CTSSP2RX7CTSKTSHR
SCHEMBL699212 0.70 TSHR (0.65) P2RX7TSHRHTTTAS1R3TAS1R1
SCHEMBL31004827 0.70 TSHR (0.65) P2RX7TSHRHTTTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007056163-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-18 WO disclosed