SCHEMBL14545327

SCHEMBL14545327

Clc1ccc(-c2ncc(O[C@H]3CCN(Cc4ccccc4)C3)nc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.46
ACHE P22303 3/20 0.45
DRD2 P14416 6/20 0.45
DRD4 P21917 6/20 0.45
DRD3 P35462 5/20 0.45
ROCK1 Q13464 5/20 0.43
ROCK2 O75116 3/20 0.43
BCHE P06276 2/20 0.43
BACE1 P56817 2/20 0.43
KCNH2 Q12809 1/20 0.43
CCR2 P41597 1/20 0.42
CHEK2 O96017 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14545335 0.94 ACHE (0.49) ACHEDRD2DRD4DRD3ROCK1
SCHEMBL14545566 0.81 ESR1 (0.43)
SCHEMBL14545603 0.79 MET (0.43) DRD4ALDH1A1
SCHEMBL4693991 0.78 PIK3CD (0.43) MCHR1KCNH2
SCHEMBL14544975 0.77 ACHE (0.55) ACHEDRD2DRD4DRD3ROCK1
SCHEMBL14545007 0.77 ACHE (0.55) ACHEDRD2DRD4DRD3ROCK1
SCHEMBL10607203 0.76 HRH3 (0.60) MCHR1ACHEROCK1ROCK2BCHE
SCHEMBL14545592 0.76 CNR1 (0.43)
Hydrochloric Acid SCHEMBL10608924 0.75 GAA (0.61) MCHR1ACHEROCK1ROCK2BCHE
SCHEMBL14545572 0.74 ACHE (0.62) MCHR1ACHEDRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070078135-A1 Substituted heteroaryl CB1 antagonists NEUROGEN CORPORATION (US) 2007-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070078135-A1 Substituted heteroaryl CB1 antagonists CNR1, CNR2, OPRL1 MCHR1 132/4885ACHE 1931/4885DRD2 110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.